SCHEMBL7871519

SCHEMBL7871519

CCCCCCCCC1C(C(=O)OCC#Cc2cccnc2)=C(C)NC(c2ccc(-n3ccnc3)cc2)=C1C(=O)OC

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.37
HTT P42858 1/20 0.35
TRPV1 Q8NER1 1/20 0.34
MAPT P10636 3/20 0.34
MAPK1 P28482 1/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
LMNA P02545 2/20 0.33
TMIGD3 P0DMS9 1/20 0.33
NPSR1 Q6W5P4 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7876069 0.89 ADORA3 (0.39) ADORA3HTTTRPV1MAPK1CYP3A4
SCHEMBL7864235 0.88 ADORA3 (0.38) ADORA3TRPV1MAPTMAPK1CYP3A4
SCHEMBL7871558 0.86 ADORA3 (0.43) ADORA3TRPV1MAPTMAPK1CYP3A4
SCHEMBL7869557 0.83 ADORA3 (0.42) ADORA3TRPV1MAPTMAPK1CYP3A4
SCHEMBL7872517 0.82 ADORA3 (0.38) ADORA3TRPV1MAPTMAPK1CYP3A4
SCHEMBL7871376 0.80 ADORA3 (0.37) ADORA3TRPV1MAPTMAPK1TMIGD3
SCHEMBL7873250 0.80 ADORA3 (0.37) ADORA3TRPV1MAPTMAPK1CYP3A4
SCHEMBL7869546 0.79 ADORA3 (0.41) ADORA3HTTTRPV1MAPTMAPK1
SCHEMBL8325950 0.79 ADORA3 (0.46) ADORA3HTTTRPV1MAPTCYP3A4
SCHEMBL7869547 0.79 ADORA3 (0.55) ADORA3HTTMAPTMAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed