SCHEMBL7876375

SCHEMBL7876375

c1ccc2cc(C3CCN(CCCOc4cccc5[nH]ccc45)CC3)ccc2c1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 12/20 0.51
SLC6A4 P31645 4/20 0.51
DRD2 P14416 2/20 0.51
DRD4 P21917 1/20 0.47
HRH3 Q9Y5N1 2/20 0.46
CHRM1 P11229 1/20 0.45
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7884092 0.97 HTR1A (0.51) HTR1ASLC6A4DRD2HRH3
SCHEMBL7881284 0.96 HRH3 (0.52) HTR1ASLC6A4DRD2HRH3
SCHEMBL7885417 0.95 HTR1A (0.54) HTR1ASLC6A4DRD2
SCHEMBL7876370 0.91 HTR1A (0.55) HTR1ASLC6A4DRD2
SCHEMBL7965634 0.87 HTR1A (0.47) HTR1ASLC6A4DRD4HRH3
SCHEMBL7887658 0.85 HTR1A (0.51) HTR1ASLC6A4
Oxalic Acid SCHEMBL7882940 0.83 ALDH1A1 (0.48) HTR1ADRD2
SCHEMBL7881145 0.83 HTR1A (0.72) HTR1ASLC6A4
SCHEMBL8871828 0.83 HTR1A (0.72) HTR1ASLC6A4
SCHEMBL6576189 0.81 HTR1A (0.62) HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6172073-B1 BENZIMIDAZOLYLOXY ALKANAMINES AS SEROTONIN REUPTAKE INHIBITORS; NICOTINE AND TOBACCO WITHDRAWAL; PSYCHOLOGICAL, EATING, BRAIN, GASTROINTESTINAL, SLEEP, AND SEXUAL DISORDERS ELI LILLY AND COMPANY 2001-01-09 US disclosed
US-5789402-A Compounds having effects on serotonin-related systems ELI LILLY COMPANY (US) 1998-08-04 US disclosed
US-5741789-A HETERO-OXY ALKANAMINES ELI LILLY AND COMPANY (US) 1998-04-21 US disclosed
US-5627196-A ANTIDEPRESSANTS AND ANTISEROTONIN AGENTS ELI LILLY AND COMPANY (US) 1997-05-06 US disclosed
US-5614523-A INDOLYLOXY COMPOUNDS ELI LILLY AND COMPANY (US) 1997-03-25 US disclosed
US-5576321-A ALKOXY-SUBSTITUTED INDOLES ELI LILLY AND COMPANY (US) 1996-11-19 US disclosed
WO-1996022290-A1 COMPOUNDS HAVING EFFECTS ON SEROTONIN-RELATED SYSTEMS ELI LILLY AND COMPANY (US) 1996-07-25 WO disclosed
EP-0722941-A2 Compounds having effects on serotonin-related systems ELI LILLY AND COMPANY (US) 1996-07-24 EP disclosed