SCHEMBL7876427

SCHEMBL7876427

CSc1ccc(-c2c(-c3ccccc3)oc3ccccc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.51
MAPT P10636 2/20 0.51
ALDH1A1 P00352 1/20 0.51
GLA P06280 1/20 0.51
GAA P10253 1/20 0.51
HPGD P15428 1/20 0.51
RAB9A P51151 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
PTGS2 P35354 5/20 0.50
PLA2G2A P14555 1/20 0.47
PLA2G4A P47712 1/20 0.47
PTGS1 P23219 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.43
DDR2 Q16832 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL592430 0.85 CA1 (0.55) KDM4EMAPTALDH1A1GAAHPGD
SCHEMBL29598541 0.83 PTGS2 (0.54) KDM4EMAPTALDH1A1GAAHPGD
SCHEMBL22954054 0.83 PTGS2 (0.54) KDM4EMAPTALDH1A1GAAHPGD
SCHEMBL22954006 0.83 PTGS2 (0.54) KDM4EMAPTALDH1A1GAAHPGD
SCHEMBL29597790 0.83 PTGS2 (0.54) KDM4EMAPTALDH1A1GAAHPGD
Ammonia Solution, Strong SCHEMBL28686299 0.83 CA1 (0.53) KDM4EMAPTALDH1A1GAAHPGD
SCHEMBL13743032 0.82 LMNA (0.56) KDM4EMAPTALDH1A1HPGDRAB9A
SCHEMBL7876432 0.79 MAPT (0.52) KDM4EMAPTALDH1A1GLAGAA
SCHEMBL6979534 0.79 RET (0.58) KDM4EMAPTALDH1A1GLAGAA
SCHEMBL7685589 0.79 MAPK14 (0.53) KDM4EMAPTALDH1A1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329421-B1 PHENYL-SUBSTITUTED BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES; NONSTEROIDAL ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA & CO. (CA) 2001-12-11 US disclosed
EP-0778834-B1 DIARYL BICYCLIC HETEROCYCLES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC (CA) 2000-01-26 EP disclosed
US-5521213-A NONSTEROID ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1996-05-28 US disclosed