SCHEMBL7876552

SCHEMBL7876552

CO[C@H]([CH]C(=O)Nc1ccccn1)C(N)=O

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.50
RAB9A P51151 8/20 0.50
PKM P14618 3/20 0.50
TP53 P04637 2/20 0.50
GAA P10253 2/20 0.49
SMN1; SMN2 Q16637 4/20 0.46
KMT2A Q03164 2/20 0.46
F2 P00734 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45
DHODH Q02127 1/20 0.44
LMNA P02545 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7876926 0.83 NPC1 (0.53) NPC1RAB9APKMGAASMN1; SMN2
SCHEMBL7877015 0.80 NPC1 (0.53) NPC1RAB9APKMGAASMN1; SMN2
SCHEMBL3890654 0.76 GAA (0.49) NPC1RAB9APKMTP53GAA
SCHEMBL9586710 0.74 NPC1 (0.56) NPC1RAB9APKMTP53GAA
SCHEMBL9586718 0.74 NPC1 (0.56) NPC1RAB9APKMTP53GAA
SCHEMBL6056798 0.73 RAB9A (0.50) NPC1RAB9APKMTP53GAA
SCHEMBL1147615 0.73 NPC1 (0.63) NPC1RAB9APKMGAASMN1; SMN2
SCHEMBL9080412 0.73 NPC1 (0.63) NPC1RAB9APKMGAASMN1; SMN2
SCHEMBL1185009 0.73 NPC1 (0.63) NPC1RAB9APKMGAASMN1; SMN2
SCHEMBL8889652 0.72 NPC1 (0.46) NPC1RAB9APKMTP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329400-B1 INHIBITION OR ANTAGONISM OF MATRIX METALLOPROTEASES, AND/OR TUMOR NECROSIS FACTOR-ALPHA; EXTRACELLULAR MATRIX DEGRADATION, INHIBITION OF SHEDDING OF CELL SURFACE PROTEIN ECTODOMAINS AND CD23 PROTEOLYSIS GLAXO WELLCOME INC. 2001-12-11 US disclosed