SCHEMBL7876584

SCHEMBL7876584

COc1ccc(-n2nc(C(F)F)cc2-c2ccc(S(C)(=O)=O)cc2)cc1F

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.73
PTGS1 P23219 10/20 0.73
ABCB11 O95342 1/20 0.73
ALDH1A1 P00352 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8073874 0.90 PTGS2 (0.70) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL7867755 0.88 PTGS2 (0.73) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL7876272 0.86 PTGS2 (0.60) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8925421 0.84 PTGS2 (0.81) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL7463018 0.84 PTGS2 (0.81) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL29593653 0.84 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL24645 0.84 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL7874468 0.84 PTGS2 (0.70) PTGS2PTGS1
SCHEMBL7878940 0.84 PTGS2 (0.60) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL6601340 0.83 PTGS2 (0.98) PTGS2PTGS1ABCB11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316485-B1 INHIBITS ACTIVITY OF CYCLOOXYGENASE-2; FOR THERAPY AND PROPHYLAXIS OF INFLAMMATION, THROMBOSIS, RHEUMATOID ARTHRITIS, ALZHEIMER'S DISEASE; AS ANALGESIC FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US claimed
US-6316485-B1 INHIBITS ACTIVITY OF CYCLOOXYGENASE-2; FOR THERAPY AND PROPHYLAXIS OF INFLAMMATION, THROMBOSIS, RHEUMATOID ARTHRITIS, ALZHEIMER'S DISEASE; AS ANALGESIC FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US disclosed
EP-1017678-A1 1,5-DIPHENYLPYRAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-07-12 EP disclosed
WO-1999015505-A1 1,5-DIPHENYLPYRAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-04-01 WO disclosed