SCHEMBL7878665

SCHEMBL7878665

CCOc1c(N)ccc(Cl)c1C(N)C(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.34
KMT2A Q03164 3/20 0.34
HTT P42858 2/20 0.34
IKBKB O14920 3/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
CYP3A4 P08684 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
NFKB1 P19838 1/20 0.33
CYP2C19 P33261 1/20 0.33
PMP22 Q01453 1/20 0.32
NLRP3 Q96P20 1/20 0.32
ALDH1A1 P00352 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7883261 0.86 MAPT (0.34) LMNAKMT2AHTTCYP3A4CYP1A2
SCHEMBL7876696 0.72 MAPT (0.34) LMNAKMT2ACYP3A4CYP1A2ALDH1A1
SCHEMBL7878669 0.72 POLB (0.41) LMNAMAPK1POLBKDM4EHPGD
SCHEMBL27637298 0.70 APP (0.40) LMNAKMT2AGRIN2DGRIN3BGRIN1
SCHEMBL27541444 0.68 MAPK14 (0.38) MAPTL3MBTL1
SCHEMBL7203924 0.66 AAK1 (0.39) LMNAKMT2AALDH1A1HSD17B10
SCHEMBL11085866 0.65 APP (0.36) LMNAKMT2AHTTCYP2D6CYP2C9
SCHEMBL27571353 0.63 MAPT (0.52) LMNAKMT2ACYP3A4CYP1A2CYP2C9
SCHEMBL29198702 0.63 SMN1; SMN2 (0.42) LMNAKMT2AGRIN2DGRIN3BGRIN1
SCHEMBL27499603 0.63 KMT2A (0.46) LMNAKMT2ACYP1A2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1244542-C Aromatic amine derivatives having NOS inhibitory effect CHUGAI PHARMACEUTICAL CO LTD (JP) 2006-03-08 CN disclosed
US-6331553-B1 INHIBITORS OF NITRIC OXIDE SYNTHASE; TREATING CEREBROVASCULAR DISEASES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-12-18 US disclosed
EP-0949242-A1 AROMATIC AMINE DERIVATIVES HAVING NOS INHIBITORY EFFECT Chugai Seiyaku Kabushiki Kaisha (JP) 1999-10-13 EP disclosed