SCHEMBL7878798

SCHEMBL7878798

O=C1N(c2ccccc2)C2(CCN(Cc3ccccc3)CC2)C1(CO)CO

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.47
OPRL1 P41146 2/20 0.47
OPRD1 P41143 2/20 0.47
OPRK1 P41145 1/20 0.47
POLB P06746 2/20 0.46
CYP3A4 P08684 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SIGMAR1 Q99720 4/20 0.45
CYP2D6 P10635 2/20 0.45
BACE1 P56817 1/20 0.45
DRD4 P21917 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM3 P20309 1/20 0.44
CCR3 P51677 1/20 0.43
GAA P10253 2/20 0.43
TSHR P16473 2/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7886600 0.99 POLB (0.48) OPRM1OPRL1OPRD1OPRK1POLB
SCHEMBL7887888 0.76 OPRM1 (0.48) OPRM1OPRL1OPRD1OPRK1POLB
Hydrochloric Acid SCHEMBL7878793 0.75 OPRM1 (0.47) OPRM1OPRL1OPRD1OPRK1POLB
SCHEMBL3004252 0.73 SIGMAR1 (0.47) OPRM1OPRL1OPRD1OPRK1POLB
SCHEMBL7887972 0.73 BACE1 (0.47) OPRM1OPRL1OPRD1OPRK1POLB
SCHEMBL7887975 0.73 BACE1 (0.47) OPRM1OPRL1OPRD1OPRK1POLB
SCHEMBL7886451 0.72 SIGMAR1 (0.52) OPRM1OPRL1OPRD1OPRK1POLB
SCHEMBL10148844 0.72 BACE1 (0.60) OPRM1OPRL1OPRD1OPRK1CYP3A4
Hydrochloric Acid SCHEMBL7883500 0.72 POLB (0.47) OPRM1OPRL1OPRD1OPRK1POLB
Hydrochloric Acid SCHEMBL7883505 0.72 POLB (0.47) OPRM1OPRL1OPRD1OPRK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970957-B1 Diaza-spiro[3,5] nonane derivatives HOFFMANN LA ROCHE (CH) 2001-08-16 EP disclosed
US-6113527-A 3,3-BIS-HYDROXYMETHYL-7-(CIS-4-ISOPROPYL-CYCLOHEXYL)-1-PHENYL -1,7-DIAZA-SPIRO-(3.5)NONANE-2-ONE, FOR EXAMPLE; AGONISTS OF THE ORPHANIN FQ (OFQ) RECEPTOR; USEFUL IN THE TREATMENT OF PSYCHIATRIC, NEUROLOGICAL AND PHYSIOLOGICAL DISORDERS HOFFMANN-LA ROCHE INC. (US) 2000-09-05 US disclosed
EP-0970957-A1 Diaza-spiro[3,5] nonane derivatives F. HOFFMANN-LA ROCHE AG (CH) 2000-01-12 EP disclosed