SCHEMBL7879488

SCHEMBL7879488

C/C(=C\c1ccccc1N)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.57
APEX1 P27695 8/20 0.44
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
NR4A2 P43354 1/20 0.40
RXRG P48443 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HTT P42858 1/20 0.40
CYP2C9 P11712 1/20 0.38
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006887 1.00 AKR1C3 (0.57) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL31666241 0.86 AKR1C3 (0.68) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL8746671 0.86 AKR1C3 (0.68) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL3893886 0.86 AKR1C3 (0.68) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL8001495 0.85 AKR1C3 (0.38) AKR1C3KDM4EHTTCYP2C9GAA
SCHEMBL17846896 0.84 AKR1C3 (0.47) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL17846894 0.84 AKR1C3 (0.47) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL28192388 0.80 ALDH1A1 (0.44) AKR1C3KDM4EMAPT
SCHEMBL433478 0.80 TP53 (0.47) AKR1C3KDM4EHTTCYP2C9GAA
SCHEMBL7764991 0.80 AKR1C3 (0.61) AKR1C3APEX1RXRARXRBNR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014041362-A1 UV RADIATION CLEAVABLE COMPOUNDS UNIVERSITY OF BATH (GB) 2014-03-20 WO disclosed
US-6329546-B1 FOR INVESTIGATING THE MECHANISM OF ACTION OF A PHYSIOLOGICALLY ACTIVE AMINO ACID COMPOUND SUCH AS GLUTAMIC ACID IN AN ORGANISM LABORATORY OF MOLECULAR BIOPHOTONICS (JP) 2001-12-11 US disclosed
US-6229020-B1 REACTING N-SUCCINIMIDYL AND P-NITROPHENYL CINNAMATE DERIVATIVES WITH PHYSIOLOGICALLY ACTIVE SUBSTANCE SUCH AS AN AMINO ACID; PROTECTING AMINO OR HYDROXY GROUPS FOR ANALYSIS OF BIOLOGICAL REACTIONS BY IRRADIATION WITH LIGHT LABORATORY OF MOLECULAR BIOPHOTONICS (JP) 2001-05-08 US disclosed