SCHEMBL7879575

SCHEMBL7879575

Cc1ccc(S(=O)(=O)CCc2ccc(C(C)(C)NCC(O)Cn3ccnc3)cc2)cc1C

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.37
PKM P14618 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
CYP19A1 P11511 2/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
KDM4E B2RXH2 1/20 0.35
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9021332 0.89 ADRB1 (0.36) CYP19A1KMT2AALDH1A1LMNAKDM4E
SCHEMBL9021323 0.88 ADRB1 (0.40) MAPK1KDM4ERAB9A
SCHEMBL7879572 0.83 TSHR (0.38) TSHRCYP19A1KMT2AALDH1A1KDM4E
SCHEMBL7875252 0.76 CYP19A1 (0.48) TSHRMAPK1HTTCYP19A1KMT2A
Hydrochloric Acid SCHEMBL7877064 0.74 KMT2A (0.47) MAPK1HTTCYP19A1KMT2AALDH1A1
SCHEMBL7868666 0.74 ADRA2C (0.46) CYP19A1LMNA
SCHEMBL9021320 0.73 ADRB1 (0.41) MAPK1HTTKDM4ERAB9A
SCHEMBL7868757 0.69 IDH1 (0.38) KDM4ERAB9A
SCHEMBL7873921 0.69 MAPK1 (0.42) MAPK1HTTKMT2AKDM4ERAB9A
SCHEMBL7873770 0.69 CYP26A1 (0.51) MAPK1HTTALDH1A1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326500-B1 ANTIINFLAMMATORY AGENTS; ANTIALLERGENS ABBOTT LABORATORIES 2001-12-04 US disclosed
US-6215001-B1 ANTIINFLAMMATORY AGENTS, ANTIASTHMATICS, AND ANTIALLERGENS; SIDE EFFECT REDUCTION KNOLL AKTIENGESELLSCHAFT (DE) 2001-04-10 US disclosed
US-6031109-A Phenoxy-, phenylthio-, benzoyl-alkyleneaminoalkylene-imidazole derivatives as therapeutic agents KNOLL AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed
US-5780642-A NON-STEROIDAL ANTIINFLAMMATORY AGENT WHICH BLOCKS RELEASE OF ARACHIDONIC ACID FROM PHOSPHOLIPIDS; SIDE EFFECT REDUCTION KNOLL AKTIENGESELLSCHAFT (DE) 1998-07-14 US disclosed
WO-1995000493-A1 IMIDAZOLE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-01-05 WO disclosed