SCHEMBL7879929

SCHEMBL7879929

CCCCC1(c2ccc(F)cc2)OCC(C)(C)CO1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB2 P17787 1/20 0.36
SLC6A2 P23975 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
SLC6A3 Q01959 1/20 0.36
CHRND Q07001 1/20 0.36
SLC6A4 P31645 6/20 0.34
MMP13 P45452 1/20 0.33
HTR7 P34969 1/20 0.33
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3395753 0.86 GRIN1 (0.41) GRIN1GRIN2BCHRNA1CHRNGCHRNB1
SCHEMBL13242104 0.85 SLC6A4 (0.36) SLC6A4MMP13HTR7HPGD
SCHEMBL7885222 0.82 HDAC3 (0.33) GRIN1GRIN2B
SCHEMBL7879750 0.82 GRIN1 (0.43) GRIN1GRIN2BCHRNA1CHRNGCHRNB1
SCHEMBL4689099 0.81 HSD11B1 (0.42) GRIN1GRIN2BCHRNA1CHRNGCHRNB1
SCHEMBL28609062 0.79 SLC6A3 (0.39) GRIN1GRIN2BCHRNA1CHRNGCHRNB1
SCHEMBL4689021 0.78 GRIN1 (0.40) GRIN1GRIN2BCHRNA1CHRNGCHRNB1
SCHEMBL121021 0.77 SLC6A4 (0.37) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL11239184 0.72 CHRNA1 (0.35) GRIN1GRIN2BCHRNA1CHRNGCHRNB1
SCHEMBL11243462 0.71 CHRNA1 (0.34) GRIN1GRIN2BCHRNA1CHRNGCHRNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246331-A1 NR2B-selective NMDA-receptor antagonists Westfälische Wilhelms-Universität Münster (DE) 2010-11-03 EP disclosed
WO-2010122134-A1 NR2B-SELECTIVE NMDA-RECEPTOR ANTAGONISTS Westfälische Wilhelms Universität Münster (DE) 2010-10-28 WO disclosed