SCHEMBL7880274

SCHEMBL7880274

COC(=O)c1ccc2[nH]cc(CCCCN3CCCC(Cc4ccc(C)cc4)C3)c2c1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.55
SLC6A4 P31645 2/20 0.49
ADRA2A P08913 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7879034 0.94 HTR1A (0.55) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL7877114 0.93 NPC1 (0.49) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL7880351 0.93 HTR1A (0.54) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL7881308 0.93 ADRA2A (0.58) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL6959565 0.93 HTR1A (0.63) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL7881273 0.91 HTR1A (0.53) HTR1ASLC6A4ACHE
SCHEMBL27417126 0.88 HTR1A (0.55) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL6959865 0.88 BCHE (0.49) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL7352278 0.86 BCHE (0.47) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL7878911 0.86 CCR3 (0.49) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US disclosed