SCHEMBL6959865

SCHEMBL6959865

COC(=O)Oc1ccc2[nH]cc(CCCCN3CCCC(Cc4ccc(C)cc4)C3)c2c1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.49
ACHE P22303 1/20 0.49
ADRA2A P08913 2/20 0.47
ADRA2B P18089 2/20 0.47
ADRA2C P18825 2/20 0.47
ADRA1D P25100 2/20 0.47
ADRA1A P35348 2/20 0.47
ADRA1B P35368 2/20 0.47
HTR1A P08908 3/20 0.46
SLC6A4 P31645 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959392 0.94 ADRA2A (0.54) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL6951247 0.94 BCHE (0.42) BCHEACHEADRA2AADRA2BADRA2C
SCHEMBL6949399 0.94 ADRA2A (0.47) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL6954023 0.93 HTR1A (0.49) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL6958383 0.93 HTR1A (0.52) BCHEACHEADRA2AADRA2BADRA2C
SCHEMBL7352278 0.92 BCHE (0.47) BCHEACHEADRA2AADRA2BADRA2C
SCHEMBL7082018 0.91 HTR1A (0.48) HTR1A
SCHEMBL7880274 0.88 HTR1A (0.55) BCHEACHEADRA2AADRA2BADRA2C
SCHEMBL7350360 0.87 ADRA2A (0.54) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL6959528 0.87 CCR3 (0.46) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed