SCHEMBL7885129

SCHEMBL7885129

COc1ccc2cc(C(=O)c3ccc(C(=O)NCCNC(=O)OCc4ccccc4)c4ccccc34)ccc2c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
APP P05067 2/20 0.45
ACHE P22303 1/20 0.45
KMT2A Q03164 1/20 0.44
HPGDS O60760 1/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
KDM4E B2RXH2 1/20 0.44
TACR3 P29371 3/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NQO2 P16083 1/20 0.42
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7561449 0.87 ACHE (0.51) NPC1APPACHEHPGDSMAPT
SCHEMBL7560916 0.83 SMYD3 (0.52) NPC1RXFP1ACHEKMT2AMAPT
SCHEMBL7560685 0.81 CDC25B (0.52) NPC1KMT2AHPGDSMAPTALDH1A1
SCHEMBL7560673 0.76 KDM4E (0.60) NPC1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL24013679 0.76 SLC6A2 (0.49) NPC1APPACHEKMT2AHPGDS
SCHEMBL7558683 0.75 KDM4E (0.51) NPC1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL7560911 0.75 MTNR1A (0.48) NPC1ACHEALDH1A1SMN1; SMN2SLC6A2
SCHEMBL1896425 0.73 KMT2A (0.55) NPC1ACHEKMT2AMAPTALDH1A1
SCHEMBL25462523 0.73 KDM4E (0.58) NPC1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL28982954 0.70 RAB9A (0.58) NPC1ALDH1A1SMN1; SMN2L3MBTL1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001051095-A2 PARAMAGNETIC DOTA DERIVATIVES, PHARMACEUTICAL AGENTS CONTAINING THE SAME, METHODS FOR THE PRODUCTION THEREOF AND THEIR USE FOR THE MR IMAGING OF NECROSIS AND INFARCTION SCHERING AKTIENGESELLSCHAFT (DE) 2001-07-19 WO disclosed