SCHEMBL7887263

SCHEMBL7887263

CC(=O)c1cc(NCOCC[Si](C)(C)C)n2nccc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.41
KCNN3 Q9UGI6 8/20 0.38
PRKAB2 O43741 1/20 0.37
PRKAG1 P54619 1/20 0.37
PRKAA2 P54646 1/20 0.37
PRKAA1 Q13131 1/20 0.37
PRKAG3 Q9UGI9 1/20 0.37
PRKAG2 Q9UGJ0 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37
KCNN1 Q92952 2/20 0.37
KCNN2 Q9H2S1 2/20 0.37
CDK2 P24941 4/20 0.35
CCNE1 P24864 3/20 0.35
CCNT1 O60563 2/20 0.35
CDK9 P50750 2/20 0.35
CCNA1 P78396 2/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35
CCNA2 P20248 1/20 0.35
CCND1 P24385 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL45705 0.82 KCNN3 (0.57) PDE10AKCNN3PRKAB2PRKAG1PRKAA2
SCHEMBL7879251 0.79 KCNN3 (0.38) PDE10AKCNN3PRKAB2PRKAG1PRKAA2
SCHEMBL30183 0.78 CRHR1 (0.33) PRKAA1CDK2CCNE1CCNT1CDK9
SCHEMBL7874462 0.78 CCNT1 (0.43) CDK2CCNE1CCNT1CDK9CCNA1
SCHEMBL10209999 0.75 PDE10A (0.53) PDE10AKCNN3KCNN1KCNN2CDK2
SCHEMBL39693 0.75 PDE10A (0.50) PDE10AKCNN3KCNN1KCNN2CDK2
SCHEMBL47770 0.74 PDE10A (0.49) PDE10AKCNN3KCNN1KCNN2CDK2
SCHEMBL10210928 0.74 PDE10A (0.49) PDE10AKCNN3KCNN1KCNN2CDK2
SCHEMBL19818 0.70 PDE10A (0.41) PDE10AKCNN3PRKAB2PRKAG1PRKAA2
SCHEMBL901809 0.68 GSK3B (0.52) PDE10AKCNN3KCNN1KCNN2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118207-A1 PYRAZOLO [1, 5-A] PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS SCHERING CORPORATION (US) 2010-10-14 WO disclosed