SCHEMBL7895274

SCHEMBL7895274

CNC(=O)[C@H](CCC(=O)OC)NC(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.48
CTSS P25774 7/20 0.48
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
HDAC4 P56524 3/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC6 Q9UBN7 1/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
CAPN1 P07384 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CYP2D6 P10635 1/20 0.39
SELP P16109 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16976277 0.92 CTSK (0.49) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL25946274 0.87 CTSK (0.47) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL11166014 0.86 CTSK (0.52) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL8747641 0.86 CTSK (0.52) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL13286586 0.85 CTSK (0.56) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL31250500 0.85 CTSK (0.49) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL30483892 0.85 BMP1 (0.48) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL13159728 0.84 CTSS (0.46) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL1317487 0.84 CYP1A2 (0.49) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL6337223 0.84 PPARA (0.47) CTSKCTSSCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6180611-B1 INHIBITORS OF MATRIX METALLOPROTEINASES AND TUMOR NECROSIS FACTOR DARWIN DISCOVERY, LTD. (GB) 2001-01-30 US disclosed
US-5994312-A Peptidyl compounds DARWIN DISCOVERY, LTD. (GB) 1999-11-30 US disclosed