SCHEMBL789565

SCHEMBL789565

COc1ncc(Br)cc1NS(=O)(=O)c1cccnc1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.57
MTOR P42345 2/20 0.57
SLC40A1 Q9NP59 6/20 0.57
KEAP1 Q14145 1/20 0.52
NFE2L2 Q16236 1/20 0.52
PIK3CG P48736 3/20 0.51
PI4KA P42356 1/20 0.50
GLO1 Q04760 1/20 0.50
BRAF P15056 2/20 0.48
GAA P10253 1/20 0.48
CYP17A1 P05093 1/20 0.47
PIK3CD O00329 1/20 0.46
PIK3R1 P27986 1/20 0.46
PIK3CB P42338 1/20 0.46
CYP3A4 P08684 1/20 0.46
ALPL P05186 1/20 0.46
NAMPT P43490 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL358926 0.88 PIK3CG (0.63) PIK3CAMTORSLC40A1PIK3CGPI4KA
SCHEMBL28549695 0.87 PIK3CG (0.50) PIK3CAMTORPIK3CGPIK3CDPIK3R1
Ammonia Solution, Strong SCHEMBL28564473 0.86 PIK3CG (0.49) PIK3CAMTORPIK3CGPIK3CDPIK3R1
SCHEMBL14247567 0.83 PIK3CA (0.55) PIK3CAMTORSLC40A1KEAP1NFE2L2
SCHEMBL21513796 0.83 CCR4 (0.64) SLC40A1PIK3CGBRAFPIK3CD
SCHEMBL29969873 0.83 CCR4 (0.64) SLC40A1PIK3CGBRAFPIK3CD
SCHEMBL29969232 0.82 SLC40A1 (0.44) PIK3CAMTORSLC40A1KEAP1NFE2L2
SCHEMBL21513456 0.82 SLC40A1 (0.44) PIK3CAMTORSLC40A1KEAP1NFE2L2
SCHEMBL16551868 0.82 PIK3CA (0.55) PIK3CAMTORSLC40A1KEAP1NFE2L2
SCHEMBL22447546 0.81 CCR4 (0.59) PIK3CAMTORPIK3CGPIK3CDPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015120737-A1 SUBSTITUTED PYRIDOPYRIMIDINE COMPOUNDS, PREPARATION METHODS THEREFOR AND USES THEREOF 北大方正集团有限公司 2015-08-20 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed