SCHEMBL7896809

SCHEMBL7896809

COc1ccc(C(=O)C#N)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.59
CES1 P23141 2/20 0.59
CA1 P00915 5/20 0.57
CA2 P00918 5/20 0.57
PARP1 P09874 1/20 0.55
PARP10 Q53GL7 1/20 0.55
PARP2 Q9UGN5 1/20 0.55
PARP4 Q9UKK3 1/20 0.55
ALDH1A1 P00352 2/20 0.53
MAPT P10636 2/20 0.53
KDM4E B2RXH2 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
HPGD P15428 1/20 0.53
TSHR P16473 1/20 0.53
NFKB1 P19838 1/20 0.53
APEX1 P27695 1/20 0.53
BLM P54132 1/20 0.53
PMP22 Q01453 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11196196 0.91 F3 (0.60) ALDH1A1MAPTKDM4ECYP1A2CYP3A4
SCHEMBL11196194 0.91 F3 (0.60) ALDH1A1MAPTKDM4ECYP1A2CYP3A4
SCHEMBL11199460 0.83 KDM4E (0.64) CES2CES1ALDH1A1KDM4ECYP1A2
SCHEMBL10923878 0.83 PARP10 (0.53) PARP10PARP2PARP4ALDH1A1MAPT
SCHEMBL10719753 0.82 GSK3B (0.43) CA1CA2ALDH1A1MAPTKDM4E
SCHEMBL10920836 0.81 ALDH1A1 (0.48) CES2CES1PARP1ALDH1A1MAPT
SCHEMBL10840477 0.81 CES2 (0.61) CES2CES1CA1CA2PARP1
SCHEMBL2122823 0.79 CES2 (0.59) CES2CES1CA1CA2PARP1
SCHEMBL11468841 0.79 PARP10 (0.59) PARP10ALDH1A1MAPTKDM4ECYP1A2
SCHEMBL10897886 0.79 CES2 (0.67) CES2CES1PARP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4596885-A Process for the preparation of phenylglyoxylic acid esters BAYER AKTIENGESELLSCHAFT (DE) 1986-06-24 US claimed
US-4302583-A BY HEATING THE CORRESPONDING DIMERIC ACYL CYANIDE BAYER AKTIENGESELLSCHAFT (DE) 1981-11-24 US claimed
US-4143068-A PROCESS FOR THE PREPARATION OF ACYL CYANIDE COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 1979-03-06 US claimed
CN-117136335-A Photosensitive resin composition 味之素株式会社 2023-11-28 CN disclosed
CN-112321544-B Chiral quaternary carbon cyanide and preparation method thereof 深圳湾实验室坪山生物医药研发转化中心 2023-05-26 CN disclosed
CN-112321544-A Chiral quaternary carbon cyanide and preparation method thereof 深圳湾实验室坪山生物医药研发转化中心 2021-02-05 CN disclosed
US-9630933-B2 Method for producing 1-H-tetrazole derivative NIPPON SODA CO., LTD. (JP) 2017-04-25 US disclosed
US-9630933-B2 Method for producing 1-H-tetrazole derivative NIPPON SODA CO., LTD. (JP) 2017-04-25 US disclosed
US-20150322021-A1 METHOD FOR PRODUCING 1-H-TETRAZOLE DERIVATIVE NIPPON SODA CO., LTD. (JP) 2015-11-12 US disclosed
US-20150322021-A1 METHOD FOR PRODUCING 1-H-TETRAZOLE DERIVATIVE NIPPON SODA CO., LTD. (JP) 2015-11-12 US disclosed
US-20150158829-A1 METHOD FOR PRODUCING AZIDE COMPOUND, AND METHOD FOR PRODUCING 1-H-TETRAZOLE DERIVATIVE NIPPON SODA CO., LTD. (JP) 2015-06-11 US disclosed
EP-0005484-B1 PROCESS FOR THE PREPARATION OF ACYL CYANIDES BAYER AG (DE) 1980-12-10 EP disclosed
US-4238412-A CYANATION OF THE ANHYDRIDE BAYER AKTIENGESELLSCHAFT (DE) 1980-12-09 US disclosed
EP-0005484-A1 Process for the preparation of acyl cyanides BAYER AG (DE) 1979-11-28 EP disclosed
US-4143068-A PROCESS FOR THE PREPARATION OF ACYL CYANIDE COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 1979-03-06 US disclosed
US-4122116-A HERBICIDES DEUTSCHE GOLD- UND SILBER- SCHEIDEANSTALT VORMALS ROESSLER (DE) 1978-10-24 US disclosed
US-4108877-A REACTING ACYL HALIDE WITH COPPER CYANIDE WITH HEATING IN THE PRESENCE OF A CARBOXYLIC ACID NITRILE AND AN ORGANIC SOLVENT DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DE) 1978-08-22 US disclosed
US-4108875-A REACTING ACYL HALIDE WITH AN ALKALI METAL CYANIDE AND A COPPER(I) SALT IN THE PRESENCE OF A CARBOXYLIC ACID NITRILE WITH HEATING DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DE) 1978-08-22 US disclosed
US-4069252-A Process for the preparation of certain acyl cyanide compounds BAYER AKTIENGESELLSCHAFT (DT) 1978-01-17 US disclosed
US-3986972-A HYDROGEN PEROXIDE AMERICAN CYANAMID COMPANY (US) 1976-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150322021-A1 METHOD FOR PRODUCING 1-H-TETRAZOLE DERIVATIVE CBR1, RIF1, CBR3 CES2 2160/4885CES1 2747/4885CA1 130/4885
US-20150158829-A1 METHOD FOR PRODUCING AZIDE COMPOUND, AND METHOD FOR PRODUCING 1-H-TETRAZOLE DERIVATIVE AS3MT, MSMO1, ABL1 CES2 1018/4885CES1 3326/4885CA1 148/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.