SCHEMBL7897273

SCHEMBL7897273

CCN(CC)Cc1nc2c(O)c(Cl)cc(Cl)c2c(=O)n1CC1CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B13 Q7Z5P4 1/20 0.36
KDM4E B2RXH2 5/20 0.33
GLA P06280 5/20 0.33
GAA P10253 5/20 0.33
ALDH1A1 P00352 5/20 0.33
HPGD P15428 3/20 0.33
ERAP1 Q9NZ08 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GRIA2 P42262 2/20 0.33
GRIN2A Q12879 2/20 0.33
ATM Q13315 2/20 0.32
PIM1 P11309 2/20 0.32
PIM3 Q86V86 2/20 0.32
PIM2 Q9P1W9 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7897324 0.92 CRHR1 (0.33) HSD17B13GRIA2GRIN2APIM1PIM3
SCHEMBL7897177 0.91 HSD17B13 (0.35) HSD17B13ALDH1A1GRIA2GRIN2APIM1
SCHEMBL7899042 0.89 HSD17B13 (0.35) HSD17B13KDM4EGLAGAAALDH1A1
SCHEMBL7902745 0.87 KDM4E (0.37) HSD17B13KDM4EGLAGAAALDH1A1
SCHEMBL7896827 0.84 TSHR (0.36) KDM4EGLAGAAALDH1A1HPGD
SCHEMBL3467749 0.84 HSD17B13 (0.37) HSD17B13ALDH1A1MEN1KMT2APIM1
SCHEMBL7903480 0.84 CHEK1 (0.46) HSD17B13KDM4EALDH1A1MEN1KMT2A
SCHEMBL7906217 0.83 TP53 (0.39) HSD17B13KDM4EGLAGAAALDH1A1
SCHEMBL7896811 0.83 KDM4E (0.37) KDM4EGLAGAAALDH1A1HPGD
SCHEMBL7895830 0.83 HSD17B13 (0.36) HSD17B13PIM1PIM3PIM2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379510-B1 QUINAZOLINONE COMPOUNDS PRANA BIOTECHNOLOGY LTD (AU) 2016-10-26 EP disclosed
US-20150359796-A1 QUINAZOLINONE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED (AU) 2015-12-17 US disclosed
US-20150359796-A1 QUINAZOLINONE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED (AU) 2015-12-17 US disclosed
US-9145375-B2 Quinazolinone compounds PRANA BIOTECHNOLOGY LIMITED (AU) 2015-09-29 US disclosed
US-9145375-B2 Quinazolinone compounds PRANA BIOTECHNOLOGY LIMITED (AU) 2015-09-29 US disclosed
US-20150025072-A1 QUINAZOLINONE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED (AU) 2015-01-22 US disclosed
US-20150025072-A1 QUINAZOLINONE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED (AU) 2015-01-22 US disclosed
US-8889695-B2 Quinazolinone compounds PRANA BIOTECHNOLOGY LIMITED (AU) 2014-11-18 US disclosed
US-8889695-B2 Quinazolinone compounds PRANA BIOTECHNOLOGY LIMITED (AU) 2014-11-18 US disclosed
US-20120040980-A1 QUINAZOLINONE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED (AU) 2012-02-16 US disclosed
US-20120040980-A1 QUINAZOLINONE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED (AU) 2012-02-16 US disclosed
WO-2010071944-A1 QUINAZOLINONE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED (AU) 2010-07-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150359796-A1 QUINAZOLINONE COMPOUNDS PARK7, SNCA, NDUFV2 HSD17B13 2537/4885KDM4E 3990/4885GLA 1862/4885
US-20150025072-A1 QUINAZOLINONE COMPOUNDS PARK7, SNCA, NQO2 HSD17B13 2552/4885KDM4E 3927/4885GLA 1857/4885
US-20120040980-A1 QUINAZOLINONE COMPOUNDS PARK7, SNCA, NQO2 HSD17B13 2552/4885KDM4E 3927/4885GLA 1857/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.