SCHEMBL790039

SCHEMBL790039

CCS(=O)(=O)c1ccc(-c2cc3cc(-c4cnc(OC(C)C)c(-c5ccccc5S(N)(=O)=O)c4)ccc3nc2N)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 4/20 0.44
PIK3CG P48736 4/20 0.44
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
BACE1 P56817 1/20 0.34
ALOX5AP P20292 4/20 0.34
FEN1 P39748 4/20 0.34
MAP4K4 O95819 1/20 0.34
PRKDC P78527 1/20 0.34
ATR Q13535 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
KCNH2 Q12809 1/20 0.33
AKT1 P31749 1/20 0.33
PIK3CA P42336 1/20 0.33
F10 P00742 1/20 0.33
PTGS2 P35354 1/20 0.33
SCD O00767 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL790027 0.91 PI4KA (0.46) PI4KAPIK3CGCA12CA1CA2
SCHEMBL790940 0.85 PI4KA (0.41) PI4KAPIK3CGCA12CA1CA2
SCHEMBL791132 0.85 PI4KA (0.43) PI4KAPIK3CGCA12CA1CA2
SCHEMBL790040 0.81 PIK3CG (0.56) PI4KAPIK3CGPIK3CA
SCHEMBL791171 0.76 PIK3CG (0.54) PI4KAPIK3CGKCNH2PIK3CA
SCHEMBL789502 0.73 PIK3CG (0.59) PI4KAPIK3CGPIK3CA
SCHEMBL791172 0.73 PI4KA (0.68) PI4KAPIK3CGPIK3CA
SCHEMBL789599 0.73 PI4KA (0.52) PI4KAPIK3CGMAP4K4PRKDCATR
SCHEMBL10277282 0.73 PIK3CG (0.48) PI4KAPIK3CGKCNH2PIK3CA
SCHEMBL790314 0.73 PIK3CG (0.56) PI4KAPIK3CGPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed