SCHEMBL7900884

SCHEMBL7900884

C=C(N)c1cccc(CCCBr)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.40
PRSS1 P07477 2/20 0.40
PRSS2 P07478 2/20 0.40
PRSS3 P35030 2/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
CYP4F2 P78329 3/20 0.39
CYP4A11 Q02928 3/20 0.39
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
F10 P00742 1/20 0.36
CYP2D6 P10635 1/20 0.36
NOS3 P29474 1/20 0.36
NOS2 P35228 1/20 0.36
SPHK2 Q9NRA0 1/20 0.35
SPHK1 Q9NYA1 1/20 0.35
LMNA P02545 1/20 0.35
TDP1 Q9NUW8 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2822360 0.83 PARP1 (0.50) CYP4F2CYP4A11F10KMT2AHSD17B1
SCHEMBL4402199 0.77 TDP1 (0.46) NOS1CYP2D6NOS3NOS2LMNA
SCHEMBL9671720 0.75 TDP1 (0.44) NOS1CYP4F2CYP4A11CYP2D6NOS3
SCHEMBL19929597 0.75 KEAP1 (0.53)
SCHEMBL14207821 0.74 SMYD3 (0.44) PRSS1PRSS2PRSS3LOXL2CYP4F2
SCHEMBL2181233 0.73 LPL (0.43) NOS1CYP4F2CYP4A11TDP1KMT2A
SCHEMBL9860710 0.73 LPL (0.43) NOS1CYP4F2CYP4A11TDP1KMT2A
SCHEMBL25442753 0.72 PRSS1 (0.37) NOS1PRSS1PRSS2PRSS3LOXL2
SCHEMBL6614812 0.72 CYP4A11 (0.73) LOXL2CYP4F2CYP4A11KMT2A
SCHEMBL7899949 0.72 MAOB (0.61) NOS1LMNATDP1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097172-A1 NEW TETRAHYDROPYRAZOLO[3,4-C]ISOQUINOLIN-5-AMINE DERIVATIVES ALMIRALL, S.A. (ES) 2010-09-02 WO disclosed