SCHEMBL7901027

SCHEMBL7901027

COC(C(N)=O)C(c1ccccc1)(c1ccccc1)c1ccccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 6/20 0.42
KIF11 P52732 2/20 0.42
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
ADRA1A P35348 1/20 0.37
OPRK1 P41145 1/20 0.37
KCNH2 Q12809 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 1/20 0.34
CES1 P23141 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
CXCL8 P10145 1/20 0.33
HPGD P15428 2/20 0.32
RAB9A P51151 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
LMNA P02545 1/20 0.32
KCNA3 P22001 1/20 0.32
KCNE1 P15382 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4469931 0.83 KIF11 (0.38) KCNN4KIF11HTR2AHTR2CADRA1A
SCHEMBL618737 0.73 MAPT (0.48) KCNN4KIF11MAPTKMT2ACYP1A2
SCHEMBL1701240 0.72 KCNN4 (0.53) KCNN4KIF11HTR2AHTR2CADRA1A
SCHEMBL12264172 0.71 CASP1 (0.44) KCNN4KIF11HTR2AHTR2CADRA1A
SCHEMBL28773064 0.69 KIF11 (0.38) KCNN4KIF11HTR2AHTR2CADRA1A
SCHEMBL27824023 0.69 KCNN4 (0.53) KCNN4KIF11HTR2AHTR2CADRA1A
SCHEMBL4462667 0.68 KCNN4 (0.64) KCNN4KIF11HTR2AHTR2CADRA1A
SCHEMBL5967507 0.68 KCNN4 (0.49) KCNN4KIF11HTR2AHTR2CADRA1A
SCHEMBL3218104 0.68 KCNN4 (0.52) KCNN4KIF11HTR2AHTR2CADRA1A
SCHEMBL11849509 0.67 KCNN4 (0.51) KCNN4KIF11HTR2AHTR2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918514-A4 TRIARYL METHANE COMPOUNDS FOR SICKLE CELL DISEASE HARVARD COLLEGE (US) 2001-05-09 EP disclosed
EP-0918514-A1 TRIARYL METHANE COMPOUNDS FOR SICKLE CELL DISEASE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 1999-06-02 EP disclosed
WO-1997034589-A1 TRIARYL METHANE COMPOUNDS FOR SICKLE CELL DISEASE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 1997-09-25 WO disclosed