SCHEMBL7901828

SCHEMBL7901828

COCCCn1c(C2CCCN(C(=O)C[C@@H](Cc3ccc(-c4cnc(OC)nc4)cc3)NC(=O)OC(C)(C)C)C2)c(C)c2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 2/20 0.37
KLK5 Q9Y337 1/20 0.34
SCN9A Q15858 4/20 0.33
CNR2 P34972 2/20 0.33
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33
PADI4 Q9UM07 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
HTR4 Q13639 2/20 0.32
CYP3A4 P08684 1/20 0.32
KCNH2 Q12809 1/20 0.32
ACE P12821 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
USP30 Q70CQ3 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2788887 0.93 PROKR1 (0.39) PROKR1SCN9ACNR2HTR4CYP3A4
SCHEMBL7897503 0.91 SCN9A (0.32) KLK5SCN9AHRH2HRH1GPR119
SCHEMBL7891211 0.89 PROKR1 (0.42) PROKR1KLK5SCN9ACNR2HRH2
SCHEMBL7899697 0.89 PROKR1 (0.39) PROKR1KLK5SCN9ACNR2HRH2
SCHEMBL7902566 0.87 PROKR1 (0.38) PROKR1KLK5SCN9ACNR2HRH2
SCHEMBL2789639 0.87 PROKR1 (0.42) PROKR1SCN9ACNR2HTR4CYP3A4
SCHEMBL2814433 0.86 PROKR1 (0.39) PROKR1KLK5SCN9ACNR2HRH2
SCHEMBL2814434 0.86 PROKR1 (0.39) PROKR1KLK5SCN9ACNR2HRH2
SCHEMBL7897770 0.86 PROKR1 (0.37) PROKR1KLK5SCN9ACNR2HRH2
SCHEMBL2788344 0.86 PROKR1 (0.38) PROKR1KLK5SCN9ACNR2HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed