SCHEMBL7897503

SCHEMBL7897503

COCCCn1c(C2CCCN(C(=O)C[C@@H](Cc3ccc(-c4cnc(OC)nc4)cc3)NC(=O)OC(C)(C)C)C2)c(C)c2cccc(F)c21

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.32
GPR119 Q8TDV5 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
KLK5 Q9Y337 1/20 0.32
EEF2K O00418 1/20 0.31
HRH2 P25021 1/20 0.31
HRH1 P35367 1/20 0.31
ATM Q13315 1/20 0.31
REN P00797 4/20 0.31
CYP3A4 P08684 2/20 0.31
TP53 P04637 2/20 0.30
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30
KMT2A Q03164 1/20 0.30
CTSC P53634 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2791931 0.93 SCN9A (0.33) SCN9ARENCYP3A4ALDH1A1TSHR
SCHEMBL7901828 0.91 PROKR1 (0.37) SCN9AGPR119KLK5HRH2HRH1
SCHEMBL7898811 0.90 ALOX5AP (0.30) ALOX5APFEN1KLK5RENCYP3A4
SCHEMBL7900800 0.90 ALOX5AP (0.30) ALOX5APFEN1KLK5RENCYP3A4
SCHEMBL7905913 0.89 CACNA1B (0.35) SCN9AKLK5EEF2KHRH2HRH1
SCHEMBL7890024 0.89 KLK5 (0.36) SCN9AALOX5APFEN1KLK5HRH2
SCHEMBL2813838 0.89 KLK5 (0.36) SCN9AALOX5APFEN1KLK5HRH2
SCHEMBL2813840 0.89 KLK5 (0.36) SCN9AALOX5APFEN1KLK5HRH2
SCHEMBL7901258 0.87 PABPC1 (0.33) KLK5HRH2HRH1ATM
SCHEMBL7898847 0.87 MMP13 (0.35) KLK5ATMCYP3A4TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed