SCHEMBL7905360

SCHEMBL7905360

Cc1ccc(S(=O)(=O)n2cc(-c3ccc4c(c3)CCN4)c3cc(Br)cnc32)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.36
PIK3CD O00329 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
ENPP3 O14638 1/20 0.34
ENPP1 P22413 1/20 0.34
HTR6 P50406 1/20 0.34
BRD4 O60885 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
IDO1 P14902 2/20 0.33
RIPK3 Q9Y572 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33
IKBKB O14920 1/20 0.32
CHUK O15111 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7907052 0.89 PTPN11 (0.46) PTPN11L3MBTL1PIK3CDCA1CA2
SCHEMBL7910236 0.86 PTPN11 (0.40) PTPN11L3MBTL1PIK3CDCA1CA2
SCHEMBL12066674 0.86 PTPN11 (0.49) PTPN11L3MBTL1PIK3CDCYP11B1CYP11B2
SCHEMBL7907976 0.85 PTPN11 (0.50) PTPN11L3MBTL1PIK3CDCYP11B1CYP11B2
SCHEMBL31396616 0.84 PTPN11 (0.53) PTPN11L3MBTL1CA1CA2ENPP3
SCHEMBL12066665 0.83 MAP3K11 (0.47) PTPN11PIK3CDIDO1IKBKBCHUK
SCHEMBL12066045 0.82 PTPN11 (0.47) PTPN11HTR6BRD4
SCHEMBL31344454 0.80 PTPN11 (0.50) PTPN11L3MBTL1ENPP3ENPP1MEN1
SCHEMBL28503544 0.80 PTPN11 (0.44) PTPN11L3MBTL1CYP11B1CYP11B2ENPP3
SCHEMBL31396515 0.80 PTPN11 (0.47) PTPN11L3MBTL1PIK3CDCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149950-A2 BICYCLIC HETEROARYL KINASE INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2011-12-01 WO disclosed
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed