SCHEMBL7910236

SCHEMBL7910236

Cc1ccc(S(=O)(=O)n2cc(-c3ccc4c(c3)CCN4)c3nc(Br)cnc32)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.40
PIK3CD O00329 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
IDO1 P14902 2/20 0.33
RIPK3 Q9Y572 1/20 0.33
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
MAPT P10636 1/20 0.32
RECQL P46063 1/20 0.32
JAK2 O60674 1/20 0.32
JAK3 P52333 1/20 0.32
IKBKB O14920 1/20 0.32
CHUK O15111 1/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7905360 0.86 PTPN11 (0.46) PTPN11PIK3CDCA1CA2L3MBTL1
SCHEMBL7907052 0.83 PTPN11 (0.46) PTPN11PIK3CDCA1CA2L3MBTL1
SCHEMBL12066674 0.80 PTPN11 (0.49) PTPN11PIK3CDL3MBTL1CYP11B1CYP11B2
SCHEMBL7907976 0.79 PTPN11 (0.50) PTPN11PIK3CDL3MBTL1CYP11B1CYP11B2
SCHEMBL720829 0.79 TGFBR1 (0.41) PTPN11CA1CA2L3MBTL1MEN1
SCHEMBL28706993 0.78 PTPN11 (0.41) PTPN11CA1CA2L3MBTL1MEN1
SCHEMBL12066665 0.77 MAP3K11 (0.47) PTPN11PIK3CDIDO1IKBKBCHUK
SCHEMBL28712257 0.77 L3MBTL1 (0.42) PTPN11CA1CA2L3MBTL1MEN1
SCHEMBL12066045 0.76 PTPN11 (0.47) PTPN11BRD4
SCHEMBL30641868 0.76 L3MBTL1 (0.39) PTPN11L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149950-A2 BICYCLIC HETEROARYL KINASE INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2011-12-01 WO disclosed
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed