SCHEMBL7906168

SCHEMBL7906168

CCN(c1ccccc1S)N(C)C

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.34
HTR2A P28223 1/20 0.30
HRH1 P35367 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4975474 0.78 SIGMAR1 (0.36) SIGMAR1HTR2AHRH1LMNA
SCHEMBL4613507 0.76 TSHR (0.39) SIGMAR1LMNA
SCHEMBL2464159 0.75 SIGMAR1 (0.31) SIGMAR1
SCHEMBL3184970 0.72 MAPT (0.44) HTR2AHRH1LMNA
SCHEMBL22738465 0.71 DRD3 (0.37) SIGMAR1HTR2AHRH1
SCHEMBL27957024 0.71 TSHR (0.41) LMNA
Benzene SCHEMBL28133117 0.70 ALDH1A1 (0.43) HTR2AHRH1LMNA
SCHEMBL18837041 0.69 MAPT (0.37) SIGMAR1HTR2AHRH1LMNA
SCHEMBL24685224 0.69 TSHR (0.45)
SCHEMBL16304006 0.68 ACHE (0.38) SIGMAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0343714-B1 Phenylglycidate stereoisomers, conversion products thereof with e.g. 2-nitrothiophenol and preparation of diltiazem DSM NV (NL) 1994-11-02 EP claimed
EP-0343714-A1 Phenylglycidate stereoisomers, conversion products thereof with e.g. 2-nitrothiophenol and preparation of diltiazem DSM N.V. (NL) 1989-11-29 EP claimed
US-6197953-B1 ESTER INTERCHANGE, CRYSTALLIZATION, ISOMERIZATION; PREPARING 1,5-BENZOTHIAZEPINE DERIVATIVES TANABE SEIYAKU CO., LTD. (JP) 2001-03-06 US disclosed
US-5998637-A CRYSTALLIZATION; SEPARATION TANABE SEIYAKU CO., LTD. (JP) 1999-12-07 US disclosed
EP-0861834-A1 Process for preparing optically active trans-3-substituted glycidic acid ester TANABE SEIYAKU CO., LTD. (JP) 1998-09-02 EP disclosed
EP-0343714-A1 Phenylglycidate stereoisomers, conversion products thereof with e.g. 2-nitrothiophenol and preparation of diltiazem DSM N.V. (NL) 1989-11-29 EP disclosed