SCHEMBL7907888

SCHEMBL7907888

CCN(CC)c1nc2c(c(-c3ccc(N)cc3)n1)CCN(Cc1ccccc1)C2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
BRS3 P32247 4/20 0.41
C5AR1 P21730 1/20 0.40
PARP1 P09874 1/20 0.39
TNKS2 Q9H2K2 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
DHFR P00374 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
LIMK1 P53667 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2341888 0.91 HTR2A (0.53) KMT2AMEN1HTR2AHTR2CHTR2B
SCHEMBL2336671 0.90 NPSR1 (0.44) HTR2AHTR2CHTR2BALDH1A1
SCHEMBL2341806 0.88 CLPP (0.46) HTR2AHTR2CHTR2BC5AR1
SCHEMBL2333354 0.87 KDM4E (0.45) KMT2AMEN1HTR2AHTR2CHTR2B
SCHEMBL2334932 0.81 C5AR1 (0.43) KMT2AMEN1BRS3C5AR1PARP1
SCHEMBL16034465 0.77 KMT2A (0.53) KMT2AMEN1BRS3C5AR1PARP1
SCHEMBL183618 0.75 P2RX7 (0.53) KMT2AMEN1C5AR1PARP1TNKS2
Hydrochloric Acid SCHEMBL6298078 0.74 P2RX7 (0.52) KMT2AMEN1C5AR1PARP1TNKS2
SCHEMBL22720571 0.74 KMT2A (0.48) KMT2AMEN1C5AR1PARP1TNKS2
SCHEMBL4147065 0.74 C5AR1 (0.57) KMT2AMEN1C5AR1PARP1TNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010053825-A1 2-AMINOPYRIMIDINE COMPOUNDS AS SEROTONIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2010-05-14 WO disclosed