SCHEMBL7907940

SCHEMBL7907940

COC(=O)CCNC(=O)c1cccc(NC(=O)N2CCN(C(=N)N)CC2)c1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.43
NAMPT P43490 2/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8382230 0.95 CA12 (0.46) NPC1RAB9AMAPTHTTNAMPT
SCHEMBL7913448 0.91 GAA (0.45) GAANAMPT
SCHEMBL8384540 0.90 NPC1 (0.46) NPC1RAB9AMAPTHTT
SCHEMBL7909721 0.89 POLB (0.46) NPC1RAB9AGAAMAPTHTT
SCHEMBL7913440 0.88 ALDH1A1 (0.49) GAAMAPT
SCHEMBL7913458 0.88 SMN1; SMN2 (0.52) GAAMAPTHTT
SCHEMBL8381689 0.84 EPHX2 (0.53) NPC1RAB9AMAPTHTTNAMPT
SCHEMBL7913438 0.82 GAA (0.43) GAAHTT
SCHEMBL8386238 0.82 HTT (0.43) RAB9AHTTNAMPT
SCHEMBL8384343 0.82 POLB (0.48) NPC1RAB9AMAPTHTTNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608759-B1 Piperazine derivatives MERCK PATENT GMBH (DE) 2001-08-22 EP disclosed
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed
EP-0608759-A2 Piperazinderivatives MERCK PATENT GmbH (DE) 1994-08-03 EP disclosed