SCHEMBL7913448

SCHEMBL7913448

COC(=O)CCNC(=O)c1cccc(NC(=O)CNC(=O)N2CCN(C(=N)N)CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.45
ALDH1A1 P00352 2/20 0.40
SMYD3 Q9H7B4 1/20 0.40
KMT2A Q03164 2/20 0.39
PARP1 P09874 1/20 0.39
PARP10 Q53GL7 1/20 0.39
NAMPT P43490 2/20 0.39
TDP1 Q9NUW8 1/20 0.38
EPHX2 P34913 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8386238 0.92 HTT (0.43) ALDH1A1KMT2ANAMPTTDP1EPHX2
SCHEMBL7907940 0.91 NPC1 (0.45) GAANAMPT
SCHEMBL7907928 0.90 GAA (0.45) GAASMYD3KMT2ANAMPTEPHX2
SCHEMBL7913440 0.88 ALDH1A1 (0.49) GAAALDH1A1KMT2APOLB
SCHEMBL7913458 0.87 SMN1; SMN2 (0.52) GAAALDH1A1KMT2AEPHX2POLB
SCHEMBL8382230 0.87 CA12 (0.46) NAMPT
SCHEMBL8385319 0.84 NAMPT (0.47) KMT2ANAMPTEPHX2POLB
SCHEMBL8384540 0.83 NPC1 (0.46) TDP1POLB
SCHEMBL7913438 0.82 GAA (0.43) GAAALDH1A1SMYD3KMT2A
SCHEMBL8386581 0.82 FAAH (0.44) ALDH1A1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608759-B1 Piperazine derivatives MERCK PATENT GMBH (DE) 2001-08-22 EP disclosed
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed
EP-0608759-A2 Piperazinderivatives MERCK PATENT GmbH (DE) 1994-08-03 EP disclosed