SCHEMBL790844

SCHEMBL790844

Nc1nc2ccc(Br)cc2cc1C=O

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.50
ERN1 O75460 2/20 0.43
CYP2A6 P11509 3/20 0.41
HTT P42858 1/20 0.41
PABPC1 P11940 1/20 0.41
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
TLR8 Q9NR97 1/20 0.36
ADRB2 P07550 1/20 0.36
TYMS P04818 1/20 0.36
PTPN1 P18031 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22494969 0.88 BACE1 (0.50) BACE1ERN1CYP2A6HTTPABPC1
SCHEMBL13997 0.80 PSMB5 (0.47) BACE1ERN1CYP2A6HTTPABPC1
SCHEMBL8672 0.79 CYP1A2 (0.57) BACE1ERN1CYP2A6HTTKDM4E
SCHEMBL807146 0.78 TLR8 (0.55) HTTKDM4EMEN1ALDH1A1MAPT
SCHEMBL5775666 0.77 BACE1 (0.57) BACE1CYP2A6HTTPABPC1KDM4E
SCHEMBL19330294 0.75 ALDH1A1 (0.47) BACE1ERN1CYP2A6ALDH1A1CYP1A2
SCHEMBL789778 0.74 BACE1 (0.53) BACE1HTTPABPC1KDM4EMEN1
SCHEMBL21988721 0.74 BACE1 (0.53) BACE1ERN1HTTPABPC1KDM4E
SCHEMBL1632823 0.72 ERN1 (0.52) BACE1ERN1CYP2A6HTTPABPC1
SCHEMBL1162125 0.72 ERN1 (0.56) BACE1ERN1CYP2A6ALDH1A1PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed