SCHEMBL7908989

SCHEMBL7908989

Nc1ccc(-c2cnc3[nH]cc(-c4ccc5c(c4)CCN5)c3c2)cn1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 6/20 0.63
LRRK2 Q5S007 2/20 0.58
CYP3A4 P08684 2/20 0.58
CYP2D6 P10635 2/20 0.58
CYP2C9 P11712 1/20 0.58
NTRK1 P04629 5/20 0.50
PDPK1 O15530 1/20 0.50
KIT P10721 4/20 0.49
DYRK1A Q13627 3/20 0.47
CLK1 P49759 2/20 0.47
DYRK2 Q92630 2/20 0.47
DYRK1B Q9Y463 2/20 0.47
AXL P30530 1/20 0.45
CDK8 P49336 1/20 0.45
TNIK Q9UKE5 1/20 0.45
PIK3CA P42336 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7906551 0.90 KIT (0.57) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9
SCHEMBL7905041 0.90 NTRK1 (0.63) MAP3K11CYP3A4CYP2D6NTRK1KIT
SCHEMBL7907491 0.86 AXL (0.64) MAP3K11NTRK1KITAXLCDK8
SCHEMBL7910407 0.86 MAP3K11 (0.47) MAP3K11NTRK1KITDYRK1ACLK1
SCHEMBL7906025 0.84 MAP3K11 (0.69) MAP3K11NTRK1KITDYRK1ACLK1
SCHEMBL7910174 0.84 MAP3K11 (0.60) MAP3K11KITDYRK1APIK3CA
SCHEMBL7899036 0.83 KIT (0.63) MAP3K11LRRK2NTRK1KITDYRK1A
SCHEMBL12068189 0.81 DYRK1A (0.56) MAP3K11NTRK1PDPK1KITDYRK1A
SCHEMBL7906295 0.81 MAP4K1 (0.66) MAP3K11NTRK1DYRK1ACLK1DYRK2
SCHEMBL7903775 0.81 KIT (0.73) KITDYRK1APIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed