SCHEMBL7910773

SCHEMBL7910773

CCOC(=O)C1C2CCCCC2CCN1C(=O)OC

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.40
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 5/20 0.39
FKBP1A P62942 2/20 0.37
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
CHRM1 P11229 2/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 2/20 0.35
POLB P06746 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27334025 0.83 CYP3A4 (0.36) THRBATML3MBTL1ALDH1A1GAA
SCHEMBL27352660 0.82 KMT2A (0.35) L3MBTL1ALDH1A1GAAHTTKMT2A
SCHEMBL7903396 0.81 ACE (0.39) ALDH1A1POLBNPC1RAB9A
SCHEMBL7913496 0.81 EPHX1 (0.37) ALDH1A1FKBP1ANPC1RAB9A
SCHEMBL27438982 0.78 FKBP1A (0.32) FKBP1AGAAKMT2A
SCHEMBL8292058 0.78 DPP4 (0.32) GAACHRM1KMT2AMAPT
SCHEMBL3454065 0.72 ALDH1A1 (0.42) ALDH1A1HTTKMT2AMAPTPOLB
SCHEMBL27524171 0.72 GAA (0.36) THRBATML3MBTL1ALDH1A1GAA
SCHEMBL3574137 0.71 MEN1 (0.37) ALDH1A1FKBP1AGAAKMT2AMAPT
SCHEMBL13078850 0.71 MEN1 (0.37) ALDH1A1FKBP1AGAAKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6214841-B1 ANTICOAGULANTS ELI LILLY AND COMPANY 2001-04-10 US disclosed
EP-0884326-A2 Antithrombitic compound ELI LILLY AND COMPANY (US) 1998-12-16 EP disclosed
EP-0670310-B1 Bisulfite adducts of arginine aldehydes useful as thrombin inhibitors and as anticoagulants LILLY CO ELI (US) 1998-09-02 EP disclosed
EP-0670310-A1 Bisulfite adducts of arginine aldehydes useful as thrombin inhibitors and as anticoagulants ELI LILLY AND COMPANY (US) 1995-09-06 EP disclosed