SCHEMBL79109

SCHEMBL79109

CC(C)(C)c1cc(CNC(=O)CC(F)(F)F)ccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 6/20 0.50
HPGD P15428 2/20 0.47
TSHR P16473 2/20 0.44
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
TRPV1 Q8NER1 2/20 0.40
NR3C1 P04150 2/20 0.40
EPHX2 P34913 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1751254 0.83 P2RX7 (0.44) P2RX7HPGDTSHRROCK2ROCK1
SCHEMBL91285 0.82 TSHR (0.46) P2RX7HPGDTSHRSMN1; SMN2TRPV1
SCHEMBL1750533 0.81 ERCC1 (0.46) P2RX7HPGDTSHRSMN1; SMN2TRPV1
SCHEMBL1751145 0.78 TSHR (0.41) P2RX7HPGDTSHRSMN1; SMN2TRPV1
SCHEMBL5392945 0.76 SMN1; SMN2 (0.64) HPGDTSHRSMN1; SMN2
SCHEMBL1751252 0.76 P2RX7 (0.41) P2RX7HPGDTSHRSMN1; SMN2
SCHEMBL78590 0.76 EPHX2 (0.54) P2RX7HPGDTSHRSMN1; SMN2EPHX2
SCHEMBL7927014 0.75 P2RX7 (0.58) P2RX7ROCK2ROCK1TRPV1NR3C1
SCHEMBL3272732 0.74 P2RX7 (0.57) P2RX7
SCHEMBL22537452 0.74 P2RX7 (0.58) P2RX7TSHRROCK2ROCK1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed