SCHEMBL91285

SCHEMBL91285

CCc1cc(CNC(=O)CC(F)(F)F)ccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
ERCC1 P07992 2/20 0.45
ERCC4 Q92889 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HPGD P15428 3/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
P2RX7 Q99572 5/20 0.43
REN P00797 1/20 0.42
CYP3A4 P08684 1/20 0.42
TRPV1 Q8NER1 1/20 0.41
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1750533 0.90 ERCC1 (0.46) TSHRERCC1ERCC4SMN1; SMN2HPGD
SCHEMBL1750880 0.82 REN (0.42) TSHRERCC1ERCC4HPGDLMNA
SCHEMBL79109 0.82 P2RX7 (0.50) TSHRSMN1; SMN2HPGDP2RX7TRPV1
SCHEMBL1751252 0.82 P2RX7 (0.41) TSHRERCC1ERCC4SMN1; SMN2HPGD
SCHEMBL2636014 0.81 EPHX2 (0.47) ERCC1ERCC4P2RX7RENCYP3A4
SCHEMBL2636015 0.80 HSD11B1 (0.40) TSHRERCC1ERCC4SMN1; SMN2HPGD
SCHEMBL1751145 0.80 TSHR (0.41) TSHRERCC1ERCC4SMN1; SMN2HPGD
SCHEMBL3079767 0.78 TRPV1 (0.44) SMN1; SMN2HPGDLMNARENCYP3A4
SCHEMBL5392945 0.77 SMN1; SMN2 (0.64) TSHRSMN1; SMN2HPGDLMNAALDH1A1
SCHEMBL1750408 0.77 TSHR (0.50) TSHRERCC1ERCC4SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed