Octrizole

Octrizole

SCHEMBL7912436

CC(C)(C)CC(C)(C)c1ccc(O)c(-n2nc3ccccc3n2)c1.CC(C)(C)c1cc(-n2nc3ccc(Cl)cc3n2)c(O)c(C(C)(C)C)c1

nearest known ligand 0.40

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.40
KCNH2 Q12809 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
ESR1 P03372 1/20 0.40
TP53 P04637 1/20 0.40
PGR P06401 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
AR P10275 1/20 0.40
MAPT P10636 1/20 0.40
DRD1 P21728 1/20 0.40
PTGS1 P23219 1/20 0.40
SLC6A2 P23975 1/20 0.40
PDE4A P27815 1/20 0.40
MAPK1 P28482 1/20 0.40
CASP1 P29466 1/20 0.40
SLC6A4 P31645 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Octrizole SCHEMBL8599630 0.93 NPC1 (0.45) CYP3A4KCNH2SMN1; SMN2MEN1USP2
SCHEMBL22372500 0.91 NPC1 (0.44) CYP3A4KCNH2SMN1; SMN2MEN1MAPT
SCHEMBL30157198 0.87 CYP3A4 (0.50) CYP3A4KCNH2SMN1; SMN2MEN1USP2
SCHEMBL1264030 0.87 CYP3A4 (0.50) CYP3A4KCNH2SMN1; SMN2MEN1USP2
Drometrizole SCHEMBL16212519 0.87 NPC1 (0.56) CYP3A4SMN1; SMN2MEN1MAPTKMT2A
SCHEMBL11668139 0.86 NPC1 (0.43) CYP3A4MEN1TP53MAPTCASP1
Bumetrizole SCHEMBL3740116 0.85 NPC1 (0.50) KCNH2SMN1; SMN2MEN1KMT2ANPC1
SCHEMBL29349567 0.84 NPC1 (0.41) CYP3A4MEN1MAPTMAPK1KMT2A
SCHEMBL29241 0.84 NPC1 (0.41) CYP3A4MEN1MAPTMAPK1KMT2A
SCHEMBL30510201 0.83 CYP3A4 (0.38) CYP3A4KCNH2SMN1; SMN2MEN1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6214929-B1 FREE RADICAL POLYMERIZATION OF AN ETHYLENICALLY UNSATURATED MONOMER BASF AKTIENGESELLSCAFT (DE) 2001-04-10 US disclosed
EP-0779891-B1 NOVEL ACYLPHOSPHINE OXIDES CIBA GEIGY AG (CH) 1998-12-23 EP disclosed