SCHEMBL7913201

SCHEMBL7913201

C[C@H]1O[C@@H](n2cc(Cc3cccc(OCc4ccccc4)c3)c(N)nc2=O)[C@H](O)[C@@H]1O

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.48
MPO P05164 1/20 0.40
ADORA2A P29274 2/20 0.40
ADORA1 P30542 1/20 0.40
ADK P55263 1/20 0.40
DPYD Q12882 1/20 0.39
ADORA2B P29275 1/20 0.39
LMNA P02545 1/20 0.38
FAAH O00519 1/20 0.37
MGLL Q99685 1/20 0.37
P2RY6 Q15077 2/20 0.37
NT5E P21589 1/20 0.37
P2RY14 Q15391 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7913210 1.00 DHFR (0.48) DHFRMPOADORA2AADORA1ADK
SCHEMBL3822553 0.86 DHFR (0.45) DHFRMPODPYDFAAHMGLL
SCHEMBL3817701 0.83 DHFR (0.46) DHFRMPODPYD
SCHEMBL3818242 0.80 LMNA (0.63) DHFRADKLMNAP2RY6NT5E
SCHEMBL21130861 0.74 ADK (0.45) ADKLMNA
SCHEMBL2578281 0.74 LMNA (0.57) ADORA2AADORA1ADORA2BLMNA
SCHEMBL16631213 0.74 ADK (0.39) ADORA1ADKLMNA
SCHEMBL16631641 0.70 ADK (0.43) ADORA1ADK
SCHEMBL8008108 0.70 P2RY2 (0.54) ADORA2AADORA1DPYDADORA2B
SCHEMBL2579590 0.70 LMNA (0.46) ADORA2AADORA1ADORA2BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882734-A2 5'-Deoxy-cytidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-12-09 EP claimed
US-6211166-B1 COADMINISTERED WITH A 5-FLUOROURACIL DERIVATIVE; ANTICARCINOGENIC AGENTS HOFFMAN-LA ROCHE INC. 2001-04-03 US disclosed
US-6114520-A ANTITUMOR AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-09-05 US disclosed
EP-0882734-A2 5'-Deoxy-cytidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-12-09 EP disclosed