SCHEMBL7913355

SCHEMBL7913355

Fc1ccc(Nc2nnc(-c3ccccc3)c3ccccc23)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.66
ENPP3 O14638 6/20 0.64
NPSR1 Q6W5P4 2/20 0.64
KDM4E B2RXH2 2/20 0.60
THRB P10828 1/20 0.60
MAPT P10636 3/20 0.59
ALDH1A1 P00352 2/20 0.59
PDE5A O76074 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
CYP2C9 P11712 1/20 0.59
HPGD P15428 1/20 0.59
ALOX15 P16050 1/20 0.59
CYP2C19 P33261 1/20 0.59
PDE1A P54750 1/20 0.59
PDE1B Q01064 1/20 0.59
PDE3B Q13370 1/20 0.59
PDE1C Q14123 1/20 0.59
PDE3A Q14432 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7914924 0.94 NPSR1 (0.73) GAAENPP3NPSR1KDM4ETHRB
SCHEMBL8021598 0.89 NPSR1 (0.79) GAAENPP3NPSR1KDM4ETHRB
SCHEMBL580813 0.86 ENPP3 (0.70) GAAENPP3NPSR1KDM4ETHRB
SCHEMBL7904940 0.84 ENPP3 (0.70) GAAENPP3NPSR1KDM4ETHRB
SCHEMBL7915165 0.84 ALDH1A1 (0.72) GAAENPP3NPSR1KDM4ETHRB
SCHEMBL581896 0.84 GAA (0.91) GAAENPP3NPSR1KDM4ETHRB
SCHEMBL7915123 0.84 KDR (0.70) GAAENPP3NPSR1KDM4ETHRB
SCHEMBL7915163 0.84 ALDH1A1 (0.71) GAAENPP3NPSR1KDM4ETHRB
Hydrochloric Acid SCHEMBL580605 0.83 GAA (0.88) GAAENPP3NPSR1KDM4ETHRB
SCHEMBL7915070 0.81 NPSR1 (0.67) GAAENPP3NPSR1KDM4ETHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207666-B1 TREATING PRECANCEROUS LESIONS BY ADMINISTERING 4-PHENYLPHTHALAZINE DERIVATIVE CELL PATHWAYS, INC. 2001-03-27 US disclosed
EP-0975605-A1 PYRIDAZINE AND PHTHALAZINE DERIVATIVES, PROCESS OF THEIR PREPARATION AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2000-02-02 EP disclosed
WO-1998046574-A1 PYRIDAZINE AND PHTHALAZINE DERIVATIVES, PROCESS OF THEIR PREPARATION AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 1998-10-22 WO disclosed