SCHEMBL7913396

SCHEMBL7913396

COC(=O)C(Cc1ccc(OCC2CN(c3ccccc3C#N)C(=O)O2)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.49
GRM2 Q14416 8/20 0.43
YAP1 P46937 1/20 0.42
CTSS P25774 4/20 0.42
CTSK P43235 3/20 0.42
CTSB P07858 2/20 0.41
CTSL P07711 1/20 0.41
KLK5 Q9Y337 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HRH2 P25021 1/20 0.39
HRH1 P35367 1/20 0.39
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7229264 0.87 GRM2 (0.47) PTPN1GRM2YAP1ITGB3ITGA2B
SCHEMBL7228413 0.86 GRM2 (0.61) PTPN1GRM2YAP1
SCHEMBL7236747 0.81 GRM2 (0.49) GRM2ITGB3ITGA2B
SCHEMBL7229073 0.80 GRM2 (0.45) GRM2ITGB3ITGA2B
SCHEMBL7913397 0.80 GRM2 (0.45) GRM2
SCHEMBL7239008 0.77 ITGB3 (0.46) PTPN1GRM2ITGB3ITGA2B
SCHEMBL7229145 0.76 YAP1 (0.46) YAP1HRH2HRH1ITGB3ITGA2B
SCHEMBL7228437 0.76 YAP1 (0.42) PTPN1YAP1KLK5HDAC8HRH2
SCHEMBL7228364 0.75 YAP1 (0.48) YAP1HRH2HRH1
SCHEMBL7237702 0.74 HRH2 (0.47) YAP1HRH2HRH1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed