SCHEMBL7913422

SCHEMBL7913422

O=C(CN1CCNCC1=O)Nc1cccc(C(=O)O)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.53
CCKBR P32239 1/20 0.44
AKT1 P31749 1/20 0.44
POLB P06746 1/20 0.43
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 5/20 0.43
ALDH1A1 P00352 3/20 0.43
KMT2A Q03164 3/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
MEN1 O00255 2/20 0.43
HSD17B10 Q99714 1/20 0.43
HIF1A Q16665 1/20 0.42
EPAS1 Q99814 1/20 0.42
ESR1 P03372 1/20 0.42
MAPT P10636 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
APOBEC3G Q9HC16 1/20 0.42
ERAP1 Q9NZ08 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7909444 0.87 HTT (0.45) HTTPOLBSMN1; SMN2ALDH1A1KMT2A
SCHEMBL7909451 0.85 ITGB3 (0.53) HTTSMN1; SMN2KMT2A
SCHEMBL8382626 0.84 EPHX2 (0.48) HTTSMN1; SMN2KMT2AMEN1
SCHEMBL7909731 0.84 ITGB3 (0.43) HTTCCKBRSMN1; SMN2ALDH1A1KMT2A
SCHEMBL7907914 0.81 GAA (0.45) HTTPOLBSMN1; SMN2ALDH1A1KMT2A
SCHEMBL670624 0.78 CYP2C9 (0.55) HTTPOLBCYP2C19ALDH1A1KMT2A
SCHEMBL1441065 0.77 HTT (0.43) HTTAKT1POLBSMN1; SMN2ALDH1A1
SCHEMBL1441038 0.77 ALDH1A1 (0.50) HTTPOLBSMN1; SMN2ALDH1A1KMT2A
SCHEMBL5231943 0.76 KCNH2 (0.44) HTTPOLBCYP2C19SMN1; SMN2ALDH1A1
SCHEMBL7906618 0.76 HTT (0.49) HTTCCKBRPOLBCYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608759-B1 Piperazine derivatives MERCK PATENT GMBH (DE) 2001-08-22 EP disclosed
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed
EP-0608759-A2 Piperazinderivatives MERCK PATENT GmbH (DE) 1994-08-03 EP disclosed