SCHEMBL7909444

SCHEMBL7909444

O=C(O)CNC(=O)c1cccc(NC(=O)CN2CCNCC2=O)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.45
ITGB3 P05106 1/20 0.41
ITGA2 P17301 1/20 0.41
CHRM3 P20309 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
LMNA P02545 2/20 0.39
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
EPHX2 P34913 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
POLB P06746 1/20 0.39
ESR1 P03372 1/20 0.38
MAPT P10636 1/20 0.38
USP5 P45974 1/20 0.38
GAA P10253 1/20 0.38
NAMPT P43490 1/20 0.38
PARP1 P09874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7909451 0.90 ITGB3 (0.53) HTTITGB3ITGA2CHRM3SMN1; SMN2
SCHEMBL8382626 0.88 EPHX2 (0.48) HTTITGB3ITGA2CHRM3LMNA
SCHEMBL7913422 0.87 HTT (0.53) HTTALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL7909731 0.84 ITGB3 (0.43) HTTITGB3ITGA2CHRM3L3MBTL1
SCHEMBL7907914 0.84 GAA (0.45) HTTITGB3ITGA2CHRM3L3MBTL1
SCHEMBL7909741 0.80 F10 (0.41) HTTITGB3ITGA2LMNAALDH1A1
SCHEMBL7907920 0.79 ITGB3 (0.53) HTTITGB3L3MBTL1LMNAALDH1A1
SCHEMBL8382617 0.78 NAMPT (0.49) HTTCHRM3L3MBTL1EPHX2POLB
SCHEMBL8381170 0.78 CHRM3 (0.49) CHRM3L3MBTL1LMNAALDH1A1SMN1; SMN2
SCHEMBL8385665 0.77 POLB (0.58) HTTCHRM3LMNAALDH1A1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608759-B1 Piperazine derivatives MERCK PATENT GMBH (DE) 2001-08-22 EP disclosed
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed
EP-0608759-A2 Piperazinderivatives MERCK PATENT GmbH (DE) 1994-08-03 EP disclosed