SCHEMBL7914100

SCHEMBL7914100

C[C@H](NC(=O)C1(c2ccccc2)CCN(C(=O)C2CCN(c3ccc(C(N)=O)cn3)CC2)CC1)C1=CC=CCC1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.43
KDM1A O60341 1/20 0.37
ENPP2 Q13822 2/20 0.36
OPRM1 P35372 1/20 0.35
OPRL1 P41146 1/20 0.35
NPY1R P25929 1/20 0.35
TACR3 P29371 1/20 0.35
PRMT5 O14744 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7907478 0.91 NPY1R (0.36) HRH3NPY1RPRMT5
SCHEMBL3106981 0.87 HRH3 (0.48) HRH3KDM1AENPP2OPRM1OPRL1
SCHEMBL7909106 0.84 MAPT (0.42) NPY1R
SCHEMBL7908842 0.80 TACR1 (0.40) HRH3NPY1R
SCHEMBL7912190 0.80 CHRM4 (0.42) HRH3NPY1R
SCHEMBL13102680 0.78 NPY1R (0.44) NPY1R
SCHEMBL7909786 0.77 NAMPT (0.41) HRH3
SCHEMBL7915500 0.75 ALDH1A1 (0.42) HRH3
SCHEMBL7908933 0.74 TSHR (0.41)
SCHEMBL13092217 0.74 KMT2A (0.52) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed