SCHEMBL7915500

SCHEMBL7915500

C[C@H](NC(=O)C1(C2=CC=CCC2)CCN(C(=O)c2ccc(N3CCCCC3)nc2)CC1)C1=CC=CCC1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
ALOX15 P16050 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ADRA1A P35348 2/20 0.37
FASN P49327 7/20 0.35
HRH3 Q9Y5N1 1/20 0.35
MGLL Q99685 1/20 0.35
GRM5 P41594 4/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
TRPV4 Q9HBA0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7913727 0.87 KDM4E (0.37) ALDH1A1KDM4EPOLBADRA1ASMN1; SMN2
SCHEMBL7910233 0.80 CYP3A4 (0.34) ALDH1A1HPGDHRH3
SCHEMBL7908118 0.78 ALDH1A1 (0.45) ALDH1A1HPGDKDM4EALOX15
SCHEMBL7909786 0.77 NAMPT (0.41) ALDH1A1KDM4EALOX15HSD17B10HRH3
SCHEMBL7908933 0.77 TSHR (0.41) ALDH1A1ALOX15HSD17B10SMN1; SMN2
SCHEMBL7906027 0.76 ACACB (0.32)
SCHEMBL7909124 0.76 BDKRB1 (0.34) ALDH1A1FASNMGLL
SCHEMBL13092177 0.75 ALDH1A1 (0.47) ALDH1A1HPGDKDM4EPOLBALOX15
SCHEMBL7914100 0.75 HRH3 (0.43) HRH3
SCHEMBL7910389 0.73 HRH3 (0.36) ALDH1A1HPGDHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed