SCHEMBL7909786

SCHEMBL7909786

C[C@H](NC(=O)C1(c2ccccc2)CCN(C(=O)c2ccc(-n3ccnc3)nc2)CC1)C1=CC=CCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.41
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 1/20 0.35
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
TSHR P16473 3/20 0.34
HRH3 Q9Y5N1 1/20 0.34
ALOX15 P16050 1/20 0.34
OPRD1 P41143 2/20 0.34
OPRK1 P41145 2/20 0.34
CXCR4 P61073 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13092194 0.87 CYP1A2 (0.43) NAMPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL7912463 0.80 CA12 (0.37) NAMPTCYP3A4PDCD1CD274TSHR
SCHEMBL7902195 0.79 ABL1 (0.44) TSHRALOX15OPRD1OPRK1CA12
SCHEMBL7915828 0.78 TSHR (0.39) KDM4ETSHRALOX15CA12CA1
SCHEMBL7913727 0.78 KDM4E (0.37) NAMPTCYP3A4KMT2AKDM4ECXCR4
SCHEMBL7908933 0.78 TSHR (0.41) CYP1A2CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL7914100 0.77 HRH3 (0.43) HRH3
SCHEMBL7915500 0.77 ALDH1A1 (0.42) KDM4EHRH3ALOX15ALDH1A1HSD17B10
SCHEMBL7912461 0.77 CYP1A2 (0.47) CYP1A2CYP2D6CYP2C9KMT2AKDM4E
SCHEMBL7909508 0.76 CA12 (0.37) CYP3A4KMT2ATSHRHRH3ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed