SCHEMBL7916634

SCHEMBL7916634

NC(=O)c1ccc2cccc(-c3cncc(F)c3)c2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.45
CYP11B1 P15538 2/20 0.45
CYP11B2 P19099 2/20 0.45
CYP3A4 P08684 1/20 0.45
HPGDS O60760 1/20 0.44
MKNK1 Q9BUB5 6/20 0.43
MKNK2 Q9HBH9 6/20 0.43
CHEK2 O96017 2/20 0.43
PARP1 P09874 1/20 0.42
DYRK1A Q13627 2/20 0.41
PLK4 O00444 1/20 0.41
CHEK1 O14757 1/20 0.41
AURKA O14965 1/20 0.41
DAPK3 O43293 1/20 0.41
CDK1 P06493 1/20 0.41
PIM1 P11309 1/20 0.41
FGFR1 P11362 1/20 0.41
PRKACA P17612 1/20 0.41
FLT1 P17948 1/20 0.41
FGFR3 P22607 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16502521 0.88 HCAR2 (0.46) CYP17A1CYP11B1CYP11B2CYP3A4CHEK2
SCHEMBL16502773 0.87 HTR5A (0.48)
SCHEMBL16502517 0.84 CYP11B1 (0.47) CYP17A1CYP11B1CYP11B2CYP3A4DYRK1A
SCHEMBL578353 0.75 CHEK2 (0.55) MKNK1MKNK2CHEK2DYRK1APLK4
SCHEMBL30338453 0.74 BCAT2 (0.54) CYP11B1CYP11B2HPGDSMKNK1MKNK2
SCHEMBL16502534 0.73 HCAR2 (0.46) MKNK1MKNK2PIM1CSNK2A1PIM2
SCHEMBL7920221 0.72 MKNK1 (0.46) MKNK1MKNK2
SCHEMBL16502470 0.70 KMO (0.61) CYP17A1CYP11B1CYP11B2CYP3A4MKNK1
SCHEMBL4828417 0.70 PLAU (0.39) MKNK1MKNK2PARP1ROCK1SIRT2
SCHEMBL578771 0.70 PLK4 (0.57) MKNK2CHEK2PARP1DYRK1APLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010090304-A1 ACYLGUANIDINE DERIVATIVE アステラス製薬株式会社 (JP) 2010-08-12 WO disclosed