SCHEMBL7916780

SCHEMBL7916780

Cc1nc2c(cc1C(=O)NC(=N)N)CCCCC2COc1ccc(C(=O)NCCN(C)C)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
ALOX5 P09917 1/20 0.40
MAPT P10636 3/20 0.36
THRB P10828 1/20 0.36
TP53 P04637 1/20 0.36
PARP1 P09874 1/20 0.35
PDE4D Q08499 1/20 0.35
PDE7A Q13946 1/20 0.35
TRPV1 Q8NER1 2/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PRKD3 O94806 1/20 0.34
PRKD1 Q15139 1/20 0.34
PRKD2 Q9BZL6 1/20 0.34
DGAT1 O75907 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
SLC8A1 P32418 1/20 0.33
CDK1 P06493 1/20 0.33
CASP2 P42575 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7913187 0.87 ALDH1A1 (0.50) ALDH1A1ALOX5MAPTTHRBTP53
SCHEMBL7916783 0.79 ALDH1A1 (0.45) ALDH1A1ALOX5MAPTTHRBTP53
SCHEMBL927097 0.77 KDM4E (0.32) ALDH1A1HPGD
SCHEMBL7911386 0.77 ALOX5 (0.47) ALDH1A1ALOX5MAPTTHRBTP53
SCHEMBL926591 0.76 SLC9A1 (0.39) ALDH1A1MAPTTP53SMN1; SMN2
SCHEMBL927852 0.76 SLC9A1 (0.33)
SCHEMBL926206 0.76 SLC9A1 (0.33)
SCHEMBL926819 0.75 SLC9A1 (0.32)
SCHEMBL926208 0.75 SLC9A1 (0.32)
SCHEMBL928060 0.74 CNR1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6258829-B1 ANTIARRTHMIA AGENTS AND CARDIOVASCULAR DISORDERS TOA EIYO LTD. (JP) 2001-07-10 US disclosed
EP-0972767-A1 CYCLOALKA[b]PYRIDINE-3-CARBONYLGUANIDINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND DRUGS CONTAINING THE SAME TOA EIYO LTD. (JP) 2000-01-19 EP disclosed