SCHEMBL7916872

SCHEMBL7916872

CC(=O)c1cc(C)c(OCc2ccccc2)c(C(=O)O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.52
PTPN1 P18031 1/20 0.48
LMNA P02545 1/20 0.48
HPGD P15428 1/20 0.48
MRGPRX4 Q96LA9 1/20 0.47
PTGER1 P34995 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
MCL1 Q07820 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
RXRA P19793 1/20 0.46
RXRB P28702 1/20 0.46
RXRG P48443 1/20 0.46
GLRA1 P23415 1/20 0.45
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4784102 0.90 MAOB (0.59) MAOBPTPN1LMNAHPGDMRGPRX4
SCHEMBL7178694 0.86 SLC16A3 (0.46) MAOBMEN1KMT2AMCL1LTB4R
SCHEMBL9191607 0.83 DHODH (0.49) PTPN1LMNAHPGDMRGPRX4PTGER1
SCHEMBL27678664 0.82 PTGER1 (0.51) MAOBPTPN1LMNAHPGDMRGPRX4
SCHEMBL262646 0.82 MEN1 (0.63) PTPN1LMNAHPGDMRGPRX4PTGER1
SCHEMBL10698086 0.82 MCL1 (0.56) PTPN1LMNAHPGDMRGPRX4PTGER1
Hydrochloric Acid SCHEMBL16143479 0.81 MEN1 (0.61) PTPN1LMNAHPGDMRGPRX4PTGER1
SCHEMBL4308031 0.81 MEN1 (0.65) LMNAHPGDMRGPRX4MEN1KMT2A
SCHEMBL14856441 0.80 MAPT (0.55) MAOBPTPN1LMNAHPGDPTGER1
SCHEMBL7262183 0.80 MAOB (0.54) MAOBPTPN1LMNAHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6214879-B1 Allosteric inhibitors of pyruvate kinase VIRGINIA COMMONWEALTH UNIVERSITY 2001-04-10 US disclosed
WO-1999048490-A1 ALLOSTERIC INHIBITORS AND ACTIVATORS OF PYRUVATE KINASE ALLOS THERAPEUTICS, INC. (US) 1999-09-30 WO disclosed
US-5599974-A ALDEHYDE AND ACID CONTAINING COMPOUNDS BOND WITH VALINE, ARGININE, AND LYSINE OF HEMOGLOBIN MOLECULE TO MODIFY MOLECULE CENTER FOR INNOVATIVE TECHNOLOGY (US) 1997-02-04 US disclosed