SCHEMBL7921796

SCHEMBL7921796

CC1(C)[C@H]2C[C@@H]1C1OB([C@H](CC3CCC3)NC(=O)[C@H](Cc3ccccc3)NC(=O)c3cccnc3Oc3ccccc3)O[C@@H]1C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
PSMB5 P28074 8/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC2 Q92769 3/20 0.40
ITGB1 P05556 1/20 0.40
ITGA4 P13612 1/20 0.40
UGCG Q16739 2/20 0.40
HDAC3 O15379 2/20 0.39
HDAC8 Q9BY41 2/20 0.39
MAPK8 P45983 2/20 0.38
HDAC4 P56524 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7923404 0.87 PSEN1 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3148841 0.85 PSEN1 (0.58) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7922252 0.82 PSMB5 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL19381918 0.82 LMNA (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL19382097 0.81 F2 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL12279029 0.79 PSMB5 (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL19790136 0.79 PSMB5 (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL19381924 0.79 PSMB5 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7922394 0.79 PSMB5 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL19381917 0.79 PSMB5 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346882-B1 DERIVATIVES OF 1-AMINO-2-CYCLOBUTYLETHYLBORONIC ACID MILLENNIUM PHARM INC (US) 2017-09-20 EP disclosed
WO-2010036357-A1 DERIVATIVES OF 1-AMINO-2-CYCLOBUTYLETHYLBORONIC ACID MILLENNIUM PHARMACEUTICALS, INC. (US) 2010-04-01 WO disclosed