SCHEMBL7921972

SCHEMBL7921972

C=C(O)c1ccc2cccc(-c3sccc3C)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
CYP2A6 P11509 6/20 0.34
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
CYP1A2 P05177 3/20 0.32
CYP3A4 P08684 3/20 0.32
CYP2C19 P33261 3/20 0.32
KDM4E B2RXH2 3/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
ALDH1A1 P00352 1/20 0.32
PGR P06401 1/20 0.32
HTT P42858 1/20 0.32
RECQL P46063 1/20 0.32
F2 P00734 1/20 0.31
PLG P00747 1/20 0.31
PLAU P00749 1/20 0.31
PLAT P00750 1/20 0.31
KLK1 P06870 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16502516 0.86 MEN1 (0.48) MEN1KMT2ANPC1RAB9ACYP2C19
SCHEMBL7916768 0.84 KDM4E (0.38) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL16502515 0.81 NQO2 (0.42) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL7910683 0.78 HTR5A (0.47)
SCHEMBL7920129 0.73 TNF (0.45) MEN1KMT2ACYP1A2CYP2C19KDM4E
SCHEMBL7916763 0.72 RAB9A (0.35) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL16503550 0.71 KDM4E (0.36) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL16502518 0.70 PLA2G2D (0.44) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL7916817 0.70 AKR1C3 (0.41) MEN1KMT2ANPC1RAB9ACYP1A2
SCHEMBL7918345 0.70 CYP1A2 (0.40) MEN1KMT2ACYP2A6NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010090304-A1 ACYLGUANIDINE DERIVATIVE アステラス製薬株式会社 (JP) 2010-08-12 WO disclosed