Predicted protein targets (top 18)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | KMT2A | Q03164 | 3/20 | 0.44 |
| ▸ | TSHR | P16473 | 3/20 | 0.44 |
| ▸ | MEN1 | O00255 | 2/20 | 0.44 |
| ▸ | TIPARP | Q7Z3E1 | 2/20 | 0.44 |
| ▸ | TACR1 | P25103 | 1/20 | 0.44 |
| ▸ | SIGMAR1 | Q99720 | 2/20 | 0.43 |
| ▸ | MTOR | P42345 | 2/20 | 0.43 |
| ▸ | LMNA | P02545 | 4/20 | 0.43 |
| ▸ | ALDH1A1 | P00352 | 2/20 | 0.43 |
| ▸ | TDP1 | Q9NUW8 | 1/20 | 0.43 |
| ▸ | MAPT | P10636 | 3/20 | 0.43 |
| ▸ | ADAMTS5 | Q9UNA0 | 2/20 | 0.43 |
| ▸ | USP2 | O75604 | 2/20 | 0.42 |
| ▸ | ADAM17 | P78536 | 1/20 | 0.41 |
| ▸ | MC4R | P32245 | 1/20 | 0.41 |
| ▸ | ALOX15 | P16050 | 1/20 | 0.41 |
| ▸ | SMN1; SMN2 | Q16637 | 1/20 | 0.41 |
| ▸ | NPSR1 | Q6W5P4 | 1/20 | 0.41 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL16255766 | 0.93 | MTOR (0.48) | KMT2ATSHRMEN1TACR1MTOR | |
| SCHEMBL7923613 | 0.87 | MAPT (0.53) | KMT2ATSHRMEN1LMNAALDH1A1 | |
| SCHEMBL12139633 | 0.87 | TIPARP (0.45) | KMT2ATSHRMEN1TIPARPTACR1 | |
| SCHEMBL12141588 | 0.87 | TACR1 (0.47) | KMT2ATSHRMEN1TIPARPTACR1 | |
| SCHEMBL16255704 | 0.85 | KMT2A (0.52) | KMT2ATSHRMEN1LMNAALDH1A1 | |
| SCHEMBL16255781 | 0.82 | TSHR (0.65) | KMT2ATSHRMEN1MTORLMNA | |
| SCHEMBL16255703 | 0.82 | MTOR (0.48) | KMT2ATSHRMEN1TACR1MTOR | |
| SCHEMBL12142074 | 0.80 | MTOR (0.47) | KMT2AMEN1TIPARPTACR1MTOR | |
| SCHEMBL12139616 | 0.80 | MTOR (0.47) | TIPARPTACR1MTORMC4R | |
| SCHEMBL10259980 | 0.78 | ALDH1A1 (0.48) | KMT2ATSHRMEN1LMNAALDH1A1 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-8889706-B2 | Soluble mTOR complexes and modulators thereof | WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) | 2014-11-18 | — | — | US | disclosed |
| WO-2010044885-A2 | SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF | WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) | 2010-04-22 | — | — | WO | disclosed |