SCHEMBL7924315

SCHEMBL7924315

Cc1ccc2c(ccn2C)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.40
PRKCI P41743 1/20 0.39
DHFR P00374 1/20 0.39
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
HSD11B1 P28845 1/20 0.37
PIK3CB P42338 1/20 0.36
CYP2A6 P11509 1/20 0.36
RAB9A P51151 2/20 0.36
CCR1 P32246 1/20 0.36
CCR5 P51681 1/20 0.36
LMNA P02545 3/20 0.35
POLB P06746 1/20 0.35
CASP6 P55212 1/20 0.35
NQO2 P16083 1/20 0.34
MAPT P10636 2/20 0.34
TSHR P16473 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20660906 0.77 SMN1; SMN2 (0.39) PRKCIDHFRKDM4EALDH1A1GAA
SCHEMBL30592233 0.77 SMN1; SMN2 (0.39) PRKCIDHFRKDM4EALDH1A1GAA
SCHEMBL1097841 0.77 PIK3CB (0.47) PRKCIDHFRHSD11B1PIK3CBCYP2A6
SCHEMBL31036108 0.77 PIK3CB (0.47) PRKCIDHFRHSD11B1PIK3CBCYP2A6
SCHEMBL16417124 0.77 PRKCI (0.38) PRKCIDHFRKDM4EALDH1A1GAA
SCHEMBL16302770 0.75 EGFR (0.37) CYP1A2KDM4EALDH1A1GAARAB9A
SCHEMBL7706466 0.74 PRKCI (0.36) PRKCIDHFRKDM4EALDH1A1GAA
SCHEMBL17463068 0.74 CYP1A2 (0.36) CYP1A2KDM4EALDH1A1RAB9ALMNA
SCHEMBL23554638 0.72 CCR1 (0.41) PRKCIDHFRALDH1A1HSD11B1PIK3CB
SCHEMBL30547717 0.72 MGAM (0.47) PRKCIDHFRKDM4EALDH1A1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230192738-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-06-22 US disclosed
EP-3172214-B1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE DERIVATIVES AS CDK INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO LTD (CN) 2020-05-13 EP disclosed
US-9828373-B2 2-amino-pyrido[2,3-D]pyrimidin-7(8H)-one derivatives as CDK inhibitors and uses thereof SUNSHINE LAKE PHARMA CO., LTD. (CN) 2017-11-28 US disclosed
US-20170121323-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE DERIVATIVES AS CDK INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2017-05-04 US disclosed
US-20150045551-A1 FUSED AZOLE DERIVATIVE TAISHO PHARMACEUTICAL CO., LTD (JP) 2015-02-12 US disclosed
US-8501804-B2 Bicyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-08-06 US disclosed
US-8501804-B2 Bicyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-08-06 US disclosed
US-20120010247-A1 BICYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-01-12 US disclosed
US-20120010247-A1 BICYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-01-12 US disclosed
EP-2351743-A1 BICYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-08-03 EP disclosed
WO-2010050445-A1 BICYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2010-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010247-A1 BICYCLIC COMPOUND ACACA, CPT1B, ACACB CYP1A2 2432/4885PRKCI 902/4885DHFR 2852/4885
US-20170121323-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE DERIVATIVES AS CDK INHIBITORS AND USES THEREOF CDK6, CDK4, CDK7 CYP1A2 2108/4885PRKCI 949/4885DHFR 263/4885
US-20150045551-A1 FUSED AZOLE DERIVATIVE AVPR1B, AVPR1A, GRIN2B CYP1A2 838/4885PRKCI 1709/4885DHFR 367/4885
US-20230192738-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OPRM1, OPRD1, OXER1 CYP1A2 998/4885PRKCI 4488/4885DHFR 3501/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.